Compile Data Set for Download or QSAR
maximum 50k data
Found 48 with Last Name = 'serra' and Initial = 's'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019771(CHEMBL3286602)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019769(CHEMBL3286600)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019768(CHEMBL3286599)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute For Bioengineering Of Catalonia (Ibec)

Curated by ChEMBL
LigandPNGBDBM50601609(CHEMBL5175325)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of [3H]-pirenzepine from human recombinant M1 receptor expressed in CHO cells incubated for 60 mins by topcount scintillation counter me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019762(CHEMBL3286595)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50360811(CHEMBL1934677)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019770(CHEMBL3286601)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019763(CHEMBL3286596)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019765(CHEMBL3286597)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50146944(CHEMBL3765536)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human factor 12a using S-2302 as substrate assessed as para-nitroaniline release preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  6.56E+3nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus-infected BTI insect cells assessed as conversion of p-tyramine into p-hydroxyphenyl-ace...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50146992(CHEMBL3763881)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human factor 12a using S-2302 as substrate assessed as para-nitroaniline release preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  7.54E+3nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50146945(CHEMBL3763678)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human factor 12a using S-2302 as substrate assessed as para-nitroaniline release preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50360809(CHEMBL1934675)
Affinity DataIC50:  9.26E+3nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019783(CHEMBL3286612)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019764(CHEMBL1528603)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM23548(3-Carboxamide-coumarin deriv., 44 | 8-bromo-6-chlo...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human factor 12a using S-2302 as substrate assessed as para-nitroaniline release preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019784(CHEMBL3286613)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019778(CHEMBL3286607)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50360808(CHEMBL1934673)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019776(CHEMBL3286606)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50146947(CHEMBL3764790)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human factor 12a using S-2302 as substrate assessed as para-nitroaniline release preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019787(CHEMBL3286615)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50146946(CHEMBL3763449)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of human factor 12a using S-2302 as substrate assessed as para-nitroaniline release preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019766(CHEMBL3286598)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50360810(CHEMBL1934676)
Affinity DataIC50:  4.27E+4nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019791(CHEMBL3286619)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019790(CHEMBL3286618)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019789(CHEMBL3286617)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019788(CHEMBL3286616)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019786(CHEMBL3286614)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019782(CHEMBL3286611)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019781(CHEMBL3286610)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019780(CHEMBL3286609)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019779(CHEMBL3286608)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019775(CHEMBL3286605)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019774(CHEMBL444521)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019773(CHEMBL3286604)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019772(CHEMBL3286603)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019767(CHEMBL1542642)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019761(CHEMBL3286594)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019760(CHEMBL1521164)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019759(CHEMBL3286593)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  6.87E+4nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus-infected BTI insect cells assessed as conversion of p-tyramine into p-hydroxyphenyl-ace...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50360807(CHEMBL1917495)
Affinity DataIC50:  6.96E+4nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50241727((S)-2-amino-3-(1-methyl-1H-indol-3-yl)propanoic ac...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed