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Found 574 with Last Name = 'shaikh' and Initial = 'm'
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612155(CHEMBL5288797)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  0.350nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612156(CHEMBL5288389)
Affinity DataKi:  0.390nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  0.470nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612154(CHEMBL5286350)
Affinity DataKi:  0.960nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612152(CHEMBL5279810)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612158(CHEMBL5273629)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612166(CHEMBL5284402)
Affinity DataKi:  2.80nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612155(CHEMBL5288797)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612156(CHEMBL5288389)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612157(CHEMBL5265873)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612158(CHEMBL5273629)
Affinity DataKi:  5.90nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612163(CHEMBL5268744)
Affinity DataKi:  6.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612161(CHEMBL5273801)
Affinity DataKi:  8.80nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612163(CHEMBL5268744)
Affinity DataKi:  14nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612161(CHEMBL5273801)
Affinity DataKi:  16nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  26nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  35nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612164(CHEMBL5285561)
Affinity DataKi:  37nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612167(CHEMBL5276437)
Affinity DataKi:  41nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612166(CHEMBL5284402)
Affinity DataKi:  45nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612161(CHEMBL5273801)
Affinity DataKi:  45nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  47nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612152(CHEMBL5279810)
Affinity DataKi:  52nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612157(CHEMBL5265873)
Affinity DataKi:  54nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612165(CHEMBL5278830)
Affinity DataKi:  55nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612162(CHEMBL5280008)
Affinity DataKi:  61nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612154(CHEMBL5286350)
Affinity DataKi:  64nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612153(CHEMBL5275945)
Affinity DataKi:  65nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612169(CHEMBL5290815)
Affinity DataKi:  68nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 7(Homo sapiens (Human))TBA
LigandPNGBDBM50612168(CHEMBL5268000)
Affinity DataKi:  76nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612160(CHEMBL5289467)
Affinity DataKi:  79nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612159(CHEMBL5266341)
Affinity DataKi:  82nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612154(CHEMBL5286350)
Affinity DataKi:  91nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
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Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM234385(2-Methoxy-10-(2-N,N-Dimethylaminoethoxy)-5-Thia-4b...)
Affinity DataKi:  127nM ΔG°:  -40.9kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60–80 Ci/mmol), respectively. The ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612162(CHEMBL5280008)
Affinity DataKi:  188nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612163(CHEMBL5268744)
Affinity DataKi:  199nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612164(CHEMBL5285561)
Affinity DataKi:  229nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612155(CHEMBL5288797)
Affinity DataKi:  250nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612168(CHEMBL5268000)
Affinity DataKi:  291nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612153(CHEMBL5275945)
Affinity DataKi:  407nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612167(CHEMBL5276437)
Affinity DataKi:  410nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612165(CHEMBL5278830)
Affinity DataKi:  430nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612169(CHEMBL5290815)
Affinity DataKi:  461nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetCarbonic anhydrase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612164(CHEMBL5285561)
Affinity DataKi:  463nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
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