Affinity DataKi: 0.280nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.350nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.390nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.470nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.960nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.30nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.5nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.80nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.20nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.80nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.90nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 6.10nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 8.80nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 12nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 16nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 26nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 37nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 41nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 45nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 45nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 47nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 52nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 54nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 55nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 61nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 64nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 65nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 68nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 76nMAssay Description:Binding affinity to human CA7 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 79nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 82nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 91nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 127nM ΔG°: -40.9kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (6080 Ci/mmol), respectively. The ...More data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 199nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 229nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 250nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to human CA1 assessed as inhibition constantMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 291nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 407nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 410nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 430nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 461nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 463nMAssay Description:Binding affinity to human CA2 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info