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Found 381 with Last Name = 'shetty' and Initial = 's'
TargetEndothelin-1 receptor(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101257((1R,2S,3R)-1-Benzo[1,3]dioxol-5-yl-3-(2-carboxymet...)
Affinity DataKi:  0.430nMAssay Description:Tested for in vitro inhibition of [125I]-ET-1 binding to CHO cells expressing human Endothelin A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165019(4-(Diethylamino)-2-butynyl alpha-phenylcyclohexane...)
Affinity DataKi:  0.950nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165008((+)-(R)-2-(alpha-(2-(Diisopropylamino)ethyl)benzyl...)
Affinity DataKi:  6.91nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165019(4-(Diethylamino)-2-butynyl alpha-phenylcyclohexane...)
Affinity DataKi:  6.97nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165008((+)-(R)-2-(alpha-(2-(Diisopropylamino)ethyl)benzyl...)
Affinity DataKi:  7.07nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(RAT)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50099204(1229U91 | CHEMBL409762 | GR-231118 | Ile-Glu-Pro-D...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165012(CHEMBL192065 | Hydroxy-diphenyl-acetic acid 4-(3-a...)
Affinity DataKi:  14nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50101257((1R,2S,3R)-1-Benzo[1,3]dioxol-5-yl-3-(2-carboxymet...)
Affinity DataKi:  15nMAssay Description:Inhibition of [125I]-ET-1 binding to CHO cells expressing human Endothelin B receptor at a concentration of 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165012(CHEMBL192065 | Hydroxy-diphenyl-acetic acid 4-(3-a...)
Affinity DataKi:  31nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165010(CHEMBL192537 | Cyclohexyl-hydroxy-phenyl-acetic ac...)
Affinity DataKi:  35nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  37nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165020(Bis-(4-fluoro-phenyl)-hydroxy-acetic acid 4-(3-aza...)
Affinity DataKi:  39nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165020(Bis-(4-fluoro-phenyl)-hydroxy-acetic acid 4-(3-aza...)
Affinity DataKi:  40nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165018(2-((1R,5S)-3-3-Aza-bicyclo[3.1.0]hex-3-yl-1-phenyl...)
Affinity DataKi:  50nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165010(CHEMBL192537 | Cyclohexyl-hydroxy-phenyl-acetic ac...)
Affinity DataKi:  72nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  79nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165016(4-Methyl-2-[3-((1R,5S)-2-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  79nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165018(2-((1R,5S)-3-3-Aza-bicyclo[3.1.0]hex-3-yl-1-phenyl...)
Affinity DataKi:  105nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165022(4-Methyl-2-[3-((1R,5S)-1-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  118nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165022(4-Methyl-2-[3-((1R,5S)-1-methyl-3-aza-bicyclo[3.1....)
Affinity DataKi:  221nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165017(CHEMBL192485 | Cyclopentyl-hydroxy-phenyl-acetic a...)
Affinity DataKi:  224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165024(CHEMBL195169 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  291nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165013(CHEMBL194870 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  366nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165024(CHEMBL195169 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  639nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165013(CHEMBL194870 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  736nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165014(CHEMBL190459 | Cyclopentyl-hydroxy-(4-methoxy-phen...)
Affinity DataKi:  964nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165009((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165021(2-[3-((1R,5S)-1,5-Dimethyl-3-aza-bicyclo[3.1.0]hex...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165021(2-[3-((1R,5S)-1,5-Dimethyl-3-aza-bicyclo[3.1.0]hex...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165011((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165014(CHEMBL190459 | Cyclopentyl-hydroxy-(4-methoxy-phen...)
Affinity DataKi:  1.93E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165023(CHEMBL424832 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  2.61E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165023(CHEMBL424832 | N-[4-(3-Aza-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  3.58E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165015((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165011((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165009((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Ranbaxy Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165015((1R,5S)-3-[3-(2-Benzyloxy-5-methyl-phenyl)-3-pheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148383(US8962637, 108)
Affinity DataIC50:  1nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148373(US8962637, 98)
Affinity DataIC50:  1nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148382(US8962637, 107)
Affinity DataIC50:  1nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148297(US8962637, 17)
Affinity DataIC50:  2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148424(US8962637, 155)
Affinity DataIC50:  2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148367(US8962637, 92)
Affinity DataIC50:  2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Debiopharm

US Patent
LigandPNGBDBM148369(US8962637, 186 | US8962637, 94)
Affinity DataIC50:  2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
In DepthDetails US Patent
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