TargetEndothelin-1 receptor(Homo sapiens (Human))
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Tested for in vitro inhibition of [125I]-ET-1 binding to CHO cells expressing human Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Ki value for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 6.91nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 6.97nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 7.07nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of [125I]-ET-1 binding to CHO cells expressing human Endothelin B receptor at a concentration of 1 uMMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 221nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 224nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 291nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 366nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 639nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 736nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 964nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 1.93E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: 2.61E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataKi: 3.58E+3nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for rat Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Compounds were screened in the TR-FRET assay for JAK2 and c-Src kinase inhibition. Ultra light poly GT (Perkin Elmer) was used as the substrate for J...More data for this Ligand-Target Pair