TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Texas At Houston
Curated by ChEMBL
University Of Texas At Houston
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of MDM2 (unknown origin) assessed as activation of p53More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 128nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 128nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 198nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 202nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 223nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 256nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 309nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 375nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 514nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 730nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of IRAK4 in human THP-1 cells by cell based anti-inflammatory assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of IRAK1 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of IRAK1 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of IRAK1 (unknown origin)More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of IRAK1 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Zhejiang Hisun Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using testosterone as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair