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Found 99 with Last Name = 'shimada' and Initial = 'm'
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149846(2''-Amino-6''-(2-cyclopropylmethoxy-6-hydroxy-phen...)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149839(2''-Amino-6''-(2-cyclobutylmethoxy-6-hydroxy-pheny...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149833(2''-Amino-6''-(2-hydroxy-6-isobutoxy-phenyl)-1,2,3...)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149832(2''-Amino-6''-(2-hydroxy-6-propoxy-phenyl)-1,2,3,4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149838(2''-Amino-6''-(2-hydroxy-6-pentyloxy-phenyl)-1,2,3...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149825(2-Amino-6-(2-cyclopropylmethoxy-6-hydroxy-phenyl)-...)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149843(2''-Amino-6''-(2-benzyloxy-6-hydroxy-phenyl)-1,2,3...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149828(2-Amino-6-(2-cyclobutylmethoxy-6-hydroxy-phenyl)-1...)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149852(2''-Amino-6''-(2-ethoxy-6-hydroxy-phenyl)-1,2,3,4,...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149831(2''-Amino-6''-(2-heptyloxy-6-hydroxy-phenyl)-1,2,3...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149850(2-Amino-6-(2-butoxy-6-hydroxy-phenyl)-1'',2'',3'',...)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149837(2-Amino-6-(2-hydroxy-6-isobutoxy-phenyl)-1'',2'',3...)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149842(2''-Amino-6''-(2,6-dihydroxy-phenyl)-1,2,3,4,5,6-h...)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149812(2''-Amino-6''-phenyl-1,2,3,4,5,6-hexahydro-[3,4'']...)
Affinity DataIC50: >20nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149826(2-Amino-6-(2-hydroxy-6-pentyloxy-phenyl)-1'',2'',3...)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149840(2-Amino-6-(2-hydroxy-6-propoxy-phenyl)-1'',2'',3''...)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149806(2''-Amino-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexah...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149834(2-Amino-6-(2-hexyloxy-6-hydroxy-phenyl)-1'',2'',3'...)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149806(2''-Amino-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexah...)
Affinity DataIC50:  25nMAssay Description:Inhibition of I-kappa-B-kinase alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149806(2''-Amino-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexah...)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149835(2''-Amino-6''-(2-cyclohexylmethoxy-6-hydroxy-pheny...)
Affinity DataIC50:  26nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149836(2''-Amino-6''-(2-hydroxy-6-methoxy-phenyl)-1,2,3,4...)
Affinity DataIC50:  34nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149822(2-Amino-4-[1-amino-2-(4-fluoro-phenyl)-ethyl]-6-(2...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149830(2-Amino-6-(2-heptyloxy-6-hydroxy-phenyl)-1'',2'',3...)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149815(2-Amino-4-(1-amino-2-phenyl-ethyl)-6-(2-hydroxy-ph...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149815(2-Amino-4-(1-amino-2-phenyl-ethyl)-6-(2-hydroxy-ph...)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149818(2-Amino-4-(2-amino-ethyl)-6-(2-hydroxy-phenyl)-nic...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149819(2-Amino-4-[1-amino-2-(4-methoxy-phenyl)-ethyl]-6-(...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149851(2''-Amino-6''-(2-hydroxy-6-isopropoxy-phenyl)-1,2,...)
Affinity DataIC50:  81nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149820(2-Amino-4-(2-amino-2-phenyl-ethyl)-6-(2-hydroxy-ph...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149848(2-Amino-6-(2-benzyloxy-6-hydroxy-phenyl)-1'',2'',3...)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149841(2-Amino-6-(2-ethoxy-6-hydroxy-phenyl)-1'',2'',3'',...)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149809(2-Amino-4-(1-amino-ethyl)-6-(2-hydroxy-phenyl)-nic...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149807(2''-Amino-6''-(2-hydroxy-phenyl)-1-methyl-1,2,3,4,...)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149813(2''-Amino-5''-fluoro-6''-(2-hydroxy-phenyl)-1,2,3,...)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149824(2-Amino-4-(1-amino-2-methyl-propyl)-6-(2-hydroxy-p...)
Affinity DataIC50:  240nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149825(2-Amino-6-(2-cyclopropylmethoxy-6-hydroxy-phenyl)-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of I-kappa-B-kinase alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase beta More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149829(2-Amino-6-(2,6-dihydroxy-phenyl)-1'',2'',3'',4'',5...)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149810(2-Amino-6-(2-hydroxy-phenyl)-1'',2'',3'',4'',5'',6...)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149810(2-Amino-6-(2-hydroxy-phenyl)-1'',2'',3'',4'',5'',6...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149808(CHEMBL182312 | N-[3''-Cyano-6''-(2-hydroxy-phenyl)...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149823(2-Amino-4-(2-amino-propyl)-6-(2-hydroxy-phenyl)-ni...)
Affinity DataIC50:  470nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149821(2-Amino-4-(1-amino-pentyl)-6-(2-hydroxy-phenyl)-ni...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124307(2-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124310(CHEMBL170406 | Sodium; 4-{4-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149817(2''-Amino-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexah...)
Affinity DataIC50:  530nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50149847(2''-Amino-6''-(2-hydroxy-4-methoxy-phenyl)-1,2,3,4...)
Affinity DataIC50:  560nMAssay Description:Inhibition of recombinant human I-kappa-B-kinase beta (IKK beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124327(4-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124335(2-Amino-N-{3-[2-amino-3-cyano-6-(2-hydroxy-phenyl)...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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