Affinity DataIC50: 18nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: >20nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of I-kappa-B-kinase alphaMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of biotinylated Avi-tagged GDP-bound KRAS G12C mutant (1 to 185 residues) (unknown origin) assessed as inhibition of KRAS G12C mutant/SOS/...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of biotinylated Avi-tagged GDP-bound KRAS G12C mutant (1 to 185 residues) (unknown origin) assessed as inhibition of KRAS G12C mutant/SOS/...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of biotinylated Avi-tagged GDP-bound KRAS G12C mutant (1 to 185 residues) (unknown origin) assessed as inhibition of KRAS G12C mutant/SOS/...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216
Curated by ChEMBL
Kyoto 619-0216
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against recombinant human I-kappa-B-kinase betaMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of biotinylated Avi-tagged GDP-bound KRAS G12C mutant (1 to 185 residues) (unknown origin) assessed as inhibition of KRAS G12C mutant/SOS/...More data for this Ligand-Target Pair