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Found 17 with Last Name = 'shindo' and Initial = 'k'
TargetProtein kinase C delta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  87nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  360nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  480nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  600nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha-C1A domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  660nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma-C1A domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  730nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta-C1A domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50269602(CHEMBL448961 | cyclotheonamide E4)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50269601(CHEMBL507449 | cyclotheonamide E)
Affinity DataIC50:  16.1nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50269603(CHEMBL502059 | cyclotheonamide E5)
Affinity DataIC50:  67.9nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.530nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptideMore data for this Ligand-Target Pair
TargetProtein kinase C gamma type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to PKCgamma-C1A domain peptide using [3H]-labeled compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to PKCbeta-C1A domain peptide using [3H]-labeled compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.450nMAssay Description:Binding affinity to PKCeta-C1B domain peptide using [3H]-labeled compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to PKCalpha-C1A domain peptide using [3H]-labeled compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.810nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50077647(4-Hydroxy-7-(1-hydroxy-2-methylamino-ethyl)-3H-ben...)
Affinity DataKd:  51nMAssay Description:Compound was tested for its binding affinity to human Beta-2 adrenergic receptor by using the radioligand [3H]-CGP-12,177More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50077647(4-Hydroxy-7-(1-hydroxy-2-methylamino-ethyl)-3H-ben...)
Affinity DataKd:  120nMAssay Description:Compound was tested for its binding affinity to human Beta-1 adrenergic receptor by using the radioligand [3H]-CGP-12,177More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed