Affinity DataKi: 0.574nMAssay Description:Displacement of [33P]-S1P from human S1P5 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.626nMAssay Description:Agonist activity at human S1P5 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by E...More data for this Ligand-Target Pair
Affinity DataKi: 0.772nMAssay Description:Displacement of [33P]-S1P from human S1P2 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [33P]-S1P from human S1P4 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.45E+3nMAssay Description:Displacement of [33P]-S1P from rat S1P1 receptor after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.63E+3nMAssay Description:Displacement of [33P]-S1P from human S1P3 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 57nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.70E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.20E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.80E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 70nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 280nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.840nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.660nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.850nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.370nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.550nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair