TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL after differentiation assessed as effect on...More data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL during differentiation assessed as effect o...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL during differentiation assessed as effect o...More data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT in Japanese White rabbit liver microsomesMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of ACAT-mediated esterified cholesterol accumulation in human THP1 cells exposed to acetyl-LDL during differentiation assessed as effect o...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Kyoto Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of PTB1B using pNPP as substrate after 30 minsMore data for this Ligand-Target Pair