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Found 108 with Last Name = 'shirai' and Initial = 'r'
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147586((S)-4-{2-[(3R,7S)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  440nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147585((R)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  480nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150613(CHEMBL179992 | CHEMBL182645 | [(1R,4S,7aR)-1-(1,5-...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147582(4-{(R)-2-[(3aR,4S)-1-((1R,2R)-1,5-Dimethyl-hexyl)-...)
Affinity DataIC50:  860nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147587((S)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147583((S)-4-Methylene-3-{2-[(R)-7a-(R)-methyl-1-((R)-5-m...)
Affinity DataIC50:  890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activity; Value ranges from 0.44 uM to 0.89 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102414(5-(2,5-Dihydroxy-benzylamino)-N-hexyl-2-hydroxy-be...)
Affinity DataIC50:  900nMAssay Description:Displacement of [gamma-32P]-ATP from Epidermal growth factor receptor in A431 cell-free extractsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150613(CHEMBL179992 | CHEMBL182645 | [(1R,4S,7aR)-1-(1,5-...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150612(CHEMBL181402 | CHEMBL182548 | Phosphoric acid mono...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150608(2-[1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-i...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147585((R)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.44E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261103((Z)-2-(1-hexadecyl-2-oxoindolin-3-ylidene)acetic a...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147587((S)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.62E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261059((Z)-2-(2-oxo-1-tetradecylindolin-3-ylidene)acetic ...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150608(2-[1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-i...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147582(4-{(R)-2-[(3aR,4S)-1-((1R,2R)-1,5-Dimethyl-hexyl)-...)
Affinity DataIC50:  1.88E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261013((E)-2-(1-hexadecyl-2-oxoindolin-3-ylidene)acetic a...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147586((S)-4-{2-[(3R,7S)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.90E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290537((R)-4-((1Z,5E,7E)-(R)-11-Methoxy-8-methyl-tetradec...)
Affinity DataIC50:  2.50E+3nMAssay Description:Compound was evaluated for its anti tubulin activityMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290537((R)-4-((1Z,5E,7E)-(R)-11-Methoxy-8-methyl-tetradec...)
Affinity DataIC50:  2.50E+3nMAssay Description:Compound was tested for inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261012((E)-2-(1-dodecyl-2-oxoindolin-3-ylidene)acetic aci...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261058((Z)-2-(1-dodecyl-2-oxoindolin-3-ylidene)acetic aci...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150613(CHEMBL179992 | CHEMBL182645 | [(1R,4S,7aR)-1-(1,5-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150610(1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-inde...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150613(CHEMBL179992 | CHEMBL182645 | [(1R,4S,7aR)-1-(1,5-...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150615((1R,4S,7aR)-1-((R)-1,5-Dimethyl-hexyl)-7a-methyl-o...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  3.90E+3nMAssay Description:Evaluated for the inhibitory concentration against porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro tubulin polymerization-inhibitory activity.More data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50216141(CHEMBL61572)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro tubulin polymerization-inhibitory activity; 4-6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50038199(5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic ac...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [gamma-32P]-ATP from Epidermal growth factor receptor in A431 cell-free extractsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150610(1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-inde...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150611(CHEMBL362416 | Phosphoric acid mono-[(1R,4S,7aR)-1...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291039(2-[(4-Hydroxy-3-nitro-phenylamino)-methyl]-benzene...)
Affinity DataIC50:  5.40E+3nMAssay Description:Displacement of [gamma-32P]-ATP from Epidermal growth factor receptor in A431 cell-free extractsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50284111(2-Methoxy-5-[propyl-(3,4,5-trimethoxy-benzyl)-amin...)
Affinity DataIC50:  5.40E+3nMAssay Description:Evaluated for the inhibitory concentration against porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150612(CHEMBL181402 | CHEMBL182548 | Phosphoric acid mono...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150608(2-[1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-i...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150615((1R,4S,7aR)-1-((R)-1,5-Dimethyl-hexyl)-7a-methyl-o...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150612(CHEMBL181402 | CHEMBL182548 | Phosphoric acid mono...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150608(2-[1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-i...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50284103(5-[Butyl-(3,4,5-trimethoxy-benzyl)-amino]-2-methox...)
Affinity DataIC50:  7.50E+3nMAssay Description:Evaluated for the inhibitory concentration against porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  7.70E+3nMAssay Description:Concentration required for the inhibitory activity against human Cell division cycle 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261106(2-(1-dodecyl-1H-indol-3-yl)acetic acid | CHEMBL521...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150611(CHEMBL362416 | Phosphoric acid mono-[(1R,4S,7aR)-1...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150610(1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-inde...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087143(4-[(1R,7aR)-1-((R)-1,5-Dimethyl-hexyl)-7a-methyl-o...)
Affinity DataIC50:  9.00E+3nMAssay Description:Concentration required for the inhibitory activity against human Cell division cycle 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50341997(CHEMBL1765353 | Dysidiolide)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50341997(CHEMBL1765353 | Dysidiolide)
Affinity DataIC50:  9.40E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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