TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.18E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.21E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.48E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.61E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
Affinity DataIC50: 2.76E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.77E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.81E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
Affinity DataIC50: 2.82E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
Affinity DataIC50: 3.41E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
Affinity DataIC50: 3.79E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.51E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.59E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.91E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 5.06E+4nMAssay Description:Inhibition of c-Src using AEEEIYGEFEAKKKK substrate by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 5.07E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.28E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.29E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.61E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 5.77E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
Affinity DataIC50: 5.78E+4nMpH: 7.5 T: 2°CAssay Description:The kinase reaction was initiated with the incubation of the 2.5 µL of the reaction cocktail (0.7 nM of His6-Src kinase domain in kinase buffer)...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.81E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 5.83E+4nMAssay Description:Inhibition of c-Src using AEEEIYGEFEAKKKK substrate by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 5.84E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.84E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 6.05E+4nMAssay Description:Inhibition of c-Src using AEEEIYGEFEAKKKK substrate by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.06E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 6.21E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 6.58E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 6.66E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 7.16E+4nMAssay Description:Inhibition of c-Src using AEEEIYGEFEAKKKK substrate by fluorescence intensity assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 7.43E+4nMAssay Description:Inhibition of His6-tagged c-Src kinase domain using AEEEIYGEFEAKKKK as substrate pre-incubated for 10 mins before substrate addition measured after 3...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 7.45E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair