Compile Data Set for Download or QSAR
maximum 50k data
Found 9 with Last Name = 'shomin' and Initial = 'cd'
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363992(CHEMBL1950043)
Affinity DataKi:  2.72E+4nMAssay Description:Mixed type inhibition of human aurora A using kemptide as a substrate by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363992(CHEMBL1950043)
Affinity DataKi:  3.15E+4nMAssay Description:Non-competitive inhibition of human aurora-A using kemptide as a substrate by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363993(CHEMBL1950044)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human Aurora A assessed as inhibition of [gamma-33P]ATP incorporation into substrate after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363992(CHEMBL1950043)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human Aurora A assessed as inhibition of [gamma-33P]ATP incorporation into substrate after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363995(CHEMBL1950040)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of human Aurora A assessed as inhibition of [gamma-33P]ATP incorporation into substrate after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363996(CHEMBL1950041)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of human Aurora A assessed as inhibition of [gamma-33P]ATP incorporation into substrate after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363997(CHEMBL1950042)
Affinity DataIC50:  2.34E+5nMAssay Description:Inhibition of human Aurora A assessed as inhibition of [gamma-33P]ATP incorporation into substrate after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50363994(CHEMBL1950039)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human Aurora A assessed as inhibition of [gamma-33P]ATP incorporation into substrate after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM60927(1-anilinonaphthalene-8-sulfonic acid | 8-Anilino-1...)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to human Cdk2 by fluorescence spectroscopyMore data for this Ligand-Target Pair