Affinity DataKi: 9nMAssay Description:Binding affinity for 5-hydroxytryptamine 4 receptor in rat was determined by rat tunica muscularis mucosae assayMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity for 5-hydroxytryptamine 4 receptor in rat was determined by rat tunica muscularis mucosae assayMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity for 5-hydroxytryptamine 4 receptor in rat was determined by rat tunica muscularis mucosae assayMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor using [3H]GR-65630 as the radioligand in male rat cortical tissue More data for this Ligand-Target Pair
Affinity DataKi: 336nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor using [3H]GR-65630 as the radioligand in male rat cortical tissue More data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Concentration required for inhibition of 5-hydroxytryptamine 2 receptor using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Concentration required for inhibition of alpha-1 adrenergic receptor using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Compound was evaluated in a human neutrophil leukotriene B4 receptor binding assayMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibitory activity against RNA-dependent DNA polymerase(RDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Concentration required for inhibition of alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of beta adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of 5-hydroxytryptamine 2 receptor using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of beta adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of alpha-1 adrenergic receptor using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of alpha-1 adrenergic receptor using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of beta adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of alpha-1 adrenergic receptor using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of beta adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of 5-hydroxytryptamine 2 receptor using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for inhibition of 5-hydroxytryptamine 2 receptor using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibitory activity against TIBO-resistant HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibitory activity against TIBO-resistant HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibitory activity against RNA-dependent DNA polymerase(RDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research
Curated by ChEMBL
Medichem Research
Curated by ChEMBL
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
Affinity DataEC50: 538nMAssay Description:Effective concentration required towards 5-hydroxytryptamine 4 receptor in guinea pig striatum using [3H]GR-113808 as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 545nMAssay Description:Effective concentration required towards 5-hydroxytryptamine 4 receptor in guinea pig striatum using [3H]GR-113808 as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 262nMAssay Description:Effective concentration required towards 5-hydroxytryptamine 4 receptor in guinea pig striatum using [3H]GR-113808 as the radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 545nMAssay Description:Effective concentration required towards 5-hydroxytryptamine 4 receptor in guinea pig striatum using [3H]GR-113808 as the radioligandMore data for this Ligand-Target Pair