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Found 21 with Last Name = 'shrivastav' and Initial = 'a'
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425232(CHEMBL2314836)
Affinity DataIC50:  9.80nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50:  74nMAssay Description:Binding affinity to Y1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50:  80nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313459((Z)-4-oxo-4-(p-tolylamino)but-2-enoic acid | CHEMB...)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313460((Z)-4-oxo-4-(phenylamino)but-2-enoic acid | CHEMBL...)
Affinity DataIC50:  2.03E+5nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313458((Z)-4-(4-nitrophenylamino)-4-oxobut-2-enoic acid |...)
Affinity DataIC50:  2.46E+5nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313456((Z)-methyl 4-(3,4-dichlorophenylamino)-4-oxobut-2-...)
Affinity DataIC50:  4.32E+5nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313457((Z)-4-(2,6-dimethylphenylamino)-4-oxobut-2-enoic a...)
Affinity DataIC50:  4.34E+5nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313454((E)-4-(4-chlorophenylamino)-4-oxobut-2-enoic acid ...)
Affinity DataIC50:  1.60E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313447(CHEMBL1086414 | Methyl N-(3,4-dimethylphenyl)fumar...)
Affinity DataIC50:  2.33E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313450((E)-4-(4-nitrophenylamino)-4-oxobut-2-enoic acid |...)
Affinity DataIC50:  2.56E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313453((E)-4-(3,4-dichlorophenylamino)-4-oxobut-2-enoic a...)
Affinity DataIC50:  4.38E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313451((E)-4-(3,4-dimethylphenylamino)-4-oxobut-2-enoic a...)
Affinity DataIC50:  7.55E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313448((E)-methyl 4-(3,4-dichlorophenylamino)-4-oxobut-2-...)
Affinity DataIC50: >8.00E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313452((E)-4-oxo-4-(p-tolylamino)but-2-enoic acid | 4-oxo...)
Affinity DataIC50:  8.35E+6nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313455((Z)-methyl 4-oxo-4-(p-tolylamino)but-2-enoate | CH...)
Affinity DataIC50: >1.00E+7nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Acadia University

Curated by ChEMBL
LigandPNGBDBM50313449((E)-methyl 4-(4-chlorophenylamino)-4-oxobut-2-enoa...)
Affinity DataIC50:  4.00E+8nMAssay Description:Inhibition of human NMT expressed in Escherichia coli DH5alpha cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed