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Found 34 with Last Name = 'shulgin' and Initial = 'at'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063544(1-(6-(methylthio)naphthalen-2-yl)propan-2-amine | ...)
Affinity DataIC50:  74nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50003582((R-PIA)2-(4-Iodo-phenyl)-1-methyl-ethylamine | 2-(...)
Affinity DataIC50:  82nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50042722(2-Indan-5-yl-1-methyl-ethylamine | CHEMBL6842)
Affinity DataIC50:  82nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063547(1-Methyl-2-(4-methyl-benzo[1,3]dioxol-5-yl)-ethyla...)
Affinity DataIC50:  93nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063546(1-Methyl-2-(7-methyl-benzo[1,3]dioxol-5-yl)-ethyla...)
Affinity DataIC50:  107nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50005247((+/-)2-Benzo[1,3]dioxol-5-yl-1-methyl-ethylamine |...)
Affinity DataIC50:  266nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50005247((+/-)2-Benzo[1,3]dioxol-5-yl-1-methyl-ethylamine |...)
Affinity DataIC50:  478nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063545(1-Methyl-2-(6-methyl-benzo[1,3]dioxol-5-yl)-ethyla...)
Affinity DataIC50:  783nMAssay Description:Activity towards Serotonin transporter was determined by the ability to inhibit [3H]-5-HT uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50042722(2-Indan-5-yl-1-methyl-ethylamine | CHEMBL6842)
Affinity DataIC50:  849nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50003582((R-PIA)2-(4-Iodo-phenyl)-1-methyl-ethylamine | 2-(...)
Affinity DataIC50:  993nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063546(1-Methyl-2-(7-methyl-benzo[1,3]dioxol-5-yl)-ethyla...)
Affinity DataIC50:  1.49E+3nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063547(1-Methyl-2-(4-methyl-benzo[1,3]dioxol-5-yl)-ethyla...)
Affinity DataIC50:  1.94E+3nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063544(1-(6-(methylthio)naphthalen-2-yl)propan-2-amine | ...)
Affinity DataIC50:  2.38E+3nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50063545(1-Methyl-2-(6-methyl-benzo[1,3]dioxol-5-yl)-ethyla...)
Affinity DataIC50:  4.60E+3nMAssay Description:Compound was tested for the ability to inhibit [3H]-norepinephrine binding to Norepinephrine transporter in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50404655(CHEMBL282183)
Affinity DataKd:  2.45E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50404656(CHEMBL31787)
Affinity DataKd:  1.70E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005265((+/-)2-(2,5-Dimethoxy-4-methyl-phenyl)-1-methyl-et...)
Affinity DataKd:  75.9nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005264((+/-)2-(2,4-Dimethoxy-phenyl)-1-methyl-ethylamine ...)
Affinity DataKd:  2.51E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50091071((+/-)2-(2,6-Dimethoxy-phenyl)-1-methyl-ethylamine ...)
Affinity DataKd:  8.13E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005246(1-Phenylpropan-2-amin | 1-phenyl-2-aminopropane | ...)
Affinity DataKd:  5.37E+3nMAssay Description:Affinity against serotonergic receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50024209((+/-)2-(4-Methoxy-phenyl)-1-methyl-ethylamine | (-...)
Affinity DataKd:  6.92E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50164328((+/-)1-Methyl-2-(2,4,6-trimethoxy-phenyl)-ethylami...)
Affinity DataKd:  525nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005247((+/-)2-Benzo[1,3]dioxol-5-yl-1-methyl-ethylamine |...)
Affinity DataKd:  355nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50164323(2-(2-Bromo-4,5-dimethoxy-phenyl)-1-methyl-ethylami...)
Affinity DataKd:  1.78E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50024208((+/-)2-(2-Methoxy-phenyl)-1-methyl-ethylamine | 2-...)
Affinity DataKd:  2.88E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005253((+/-)1-Methyl-2-(2,4,5-trimethoxy-phenyl)-ethylami...)
Affinity DataKd:  155nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005251((+/-)2-(2,5-Dimethoxy-phenyl)-1-methyl-ethylamine ...)
Affinity DataKd:  148nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50404654(CHEMBL284589)
Affinity DataKd:  1.38E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50024211((+/-)2-(3-Methoxy-phenyl)-1-methyl-ethylamine | 2-...)
Affinity DataKd:  1.20E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50404653(CHEMBL30777)
Affinity DataKd:  8.51E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005257((+)-2-(4-Bromo-2,5-dimethoxy-phenyl)-1-methyl-ethy...)
Affinity DataKd:  44.7nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50024201((+/-)2-(3,4-Dimethoxy-phenyl)-1-methyl-ethylamine ...)
Affinity DataKd:  3.55E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50091080((+/-)2-(2,3-Dimethoxy-phenyl)-1-methyl-ethylamine ...)
Affinity DataKd:  2.88E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005256((+/-)1-Methyl-2-(3,4,5-trimethoxy-phenyl)-ethylami...)
Affinity DataKd:  2.51E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed