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Found 10 with Last Name = 'shuto' and Initial = 'd'
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50141551(5-[(S)-3-((S)-2-{(S)-2-[2-Amino-3-((S)-carboxyamin...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration of compound against Beta-secretase 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157441(5-((2R,3S)-3-((S)-2-((S)-2-((S)-2-amino-3-(2H-tetr...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory activity against beta-secretase 1 (BACE1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157442(5-{3-[2-((S)-2-{(S)-2-Amino-3-[((S)-oxalyl)-amino]...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory activity against beta-secretase 1 (BACE1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157439(3-((2R,3S)-3-((S)-2-((S)-2-((S)-2-amino-3-(2H-tetr...)
Affinity DataIC50:  8.20nMAssay Description:Inhibitory activity against beta-secretase 1 (BACE1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50141552(3-[(S)-3-((S)-2-{(S)-2-[2-Amino-3-((S)-carboxyamin...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration of compound against Beta-secretase 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157438(3-{3-[2-((S)-2-{(S)-2-Amino-3-[((S)-oxalyl)-amino]...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against beta-secretase 1 (BACE1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50141553(5-((2R,3S)-3-((S)-2-((S)-2-((S)-2-amino-4-carboxyb...)
Affinity DataIC50:  55nMAssay Description:Inhibitory concentration of compound against Beta-secretase 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50141550((S)-2-{(S)-2-[(S)-2-((S)-3-{(S)-2-[(S)-2-(2-Amino-...)
Affinity DataIC50:  84nMAssay Description:Inhibitory concentration of compound against Beta-secretase 1 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157440((S)-2-[(S)-2-((S)-2-{3-[2-((S)-2-{(S)-2-Amino-3-[(...)
Affinity DataIC50:  84nMAssay Description:Inhibitory activity against beta-secretase 1 (BACE1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50136233(CHEMBL406146 | HGluValLeuPnsAspAlaGluPheOH | KMI-0...)
Affinity DataIC50:  413nMAssay Description:Inhibitory activity of the compound against Beta-secretase 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed