Affinity DataKi: 1.30nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity of compound towards Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 197nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 368nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 373nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 426nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 497nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 518nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 615nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 875nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 970nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.24E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibitory activity against cytochrome P450 determined using human liver microsome upon 15 min incubation with probes substrates tolbutamide (2C9)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by ChEMBL
Aventis Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against human Potassium channel HERGMore data for this Ligand-Target Pair