TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 betaMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 9.80nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 betaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Affinity for human glucagon receptor in presence of Mg2+More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of LPS-induced p38-related TNF alpha release from human monocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Affinity for human glucagon receptor in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of c-Jun N-terminal kinase 2-beta 1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Binding affinity towards human Mitogen-activated protein kinase p38 expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 betaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Binding affinity towards human Mitogen-activated protein kinase p38 expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Binding affinity towards human Mitogen-activated protein kinase p38 expressed as IC50More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Rattus norvegicus)
Merck Research Laboratory
Curated by ChEMBL
Merck Research Laboratory
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibitory potency evaluated against rat p38 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of LPS-induced p38-related TNF alpha release from human monocytesMore data for this Ligand-Target Pair