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Found 13 with Last Name = 'siegal' and Initial = 'g'
TargetEphrin type-A receptor 4(Homo sapiens (Human))
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50359971(CHEMBL1927263)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 4(Homo sapiens (Human))
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50359970(CHEMBL1927262)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM81417(Fragment 1)
Affinity DataIC50:  7.00E+3nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 4(Homo sapiens (Human))
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50359969(CHEMBL1927261)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM41732(1-benzyl-2,5-dimethyl-pyrrole-3-carboxylic acid | ...)
Affinity DataIC50:  1.30E+4nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM50042278(7-Chloro-1H-quinoline-2,4-dione | CHEMBL112809 | F...)
Affinity DataIC50:  4.60E+4nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM81420(Fragment 6)
Affinity DataIC50:  7.00E+4nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM81418(Fragment 2)
Affinity DataIC50:  1.00E+5nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM81421(Fragment 7)
Affinity DataIC50:  1.15E+5nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM42347((2,2-dimethyl-4-oxo-3,4-dihydro-1,5-benzothiazepin...)
Affinity DataIC50:  1.68E+5nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisulfide bond formation protein B(Escherichia coli)
Leiden University

LigandPNGBDBM81419(Fragment 3)
Affinity DataIC50:  1.93E+5nMpH: 6.2 T: 2°CAssay Description:13 fragments with strong inhibition in the single concentration point assay were chose from the micelle screen for further analysis using a biochemic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50150060(CHEMBL3775692)
Affinity DataKd:  2.10E+4nMAssay Description:Binding affinity to N-terminal His-tagged PCAF (715 to 831 residues) (unknown origin) expressed in Escherichia coli Rosetta cells by isothermal titra...More data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50150068(CHEMBL3775323)
Affinity DataKd:  6.80E+3nMAssay Description:Binding affinity to N-terminal His-tagged PCAF (715 to 831 residues) (unknown origin) expressed in Escherichia coli Rosetta cells by isothermal titra...More data for this Ligand-Target Pair