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Found 121 with Last Name = 'sierra' and Initial = 'ml'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataIC50:  1nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataIC50:  1nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127221(CHEMBL289887 | {2-Methyl-4-[4-methyl-2-(4-trifluor...)
Affinity DataIC50:  3nMAssay Description:Maximum transcriptional activation of human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127223(CHEMBL37013 | {2-Methyl-4-[4-methyl-2-(4-trifluoro...)
Affinity DataIC50:  30nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127215(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-thiazo...)
Affinity DataIC50:  30nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127218(3-{2-Methyl-4-[4-methyl-2-(4-trifluoromethyl-pheny...)
Affinity DataIC50:  60nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127220(CHEMBL37495 | {4-[4-Methyl-2-(4-trifluoromethyl-ph...)
Affinity DataIC50:  90nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127224(3-{4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-oxazol...)
Affinity DataIC50:  90nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127216(CHEMBL416794 | {4-[4-Methyl-2-(4-trifluoromethyl-p...)
Affinity DataIC50:  340nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127219(CHEMBL39129 | {4-[4-Methyl-2-(4-trifluoromethyl-ph...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127217((E)-3-{2-Methyl-4-[4-methyl-2-(4-trifluoromethyl-p...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127225(4-[4-Methyl-2-(4-trifluoromethyl-phenyl)-oxazol-5-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity for human PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28699(2-(4-chlorophenoxy)-2-methylpropanoic acid | CHEMB...)
Affinity DataEC50:  5.50E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50:  3.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  5.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  1.89E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28702(2-[2-methyl-4-(2-{4-methyl-2-[4-(trifluoromethyl)p...)
Affinity DataEC50:  2.00E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28703(2-methyl-2-[4-(2-{4-methyl-2-[4-(trifluoromethyl)p...)
Affinity DataEC50:  210nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28704(2-methyl-2-[4-({4-methyl-2-[4-(trifluoromethyl)phe...)
Affinity DataEC50:  9.50E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM28705(2-methyl-2-(4-{[({4-methyl-2-[4-(trifluoromethyl)p...)
Affinity DataEC50:  70nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
LigandPNGBDBM28707(2-methyl-2-phenoxypropanoic acid, 27 | 2-methyl-2-...)
Affinity DataEC50:  240nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28708(2-methyl-2-phenoxypropanoic acid, 34 | 2-methyl-2-...)
Affinity DataEC50:  1.32E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28709(2-methyl-2-phenoxypropanoic acid, 37 | 2-methyl-2-...)
Affinity DataEC50:  110nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28710(2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazo...)
Affinity DataEC50:  5nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28711(2-methyl-2-phenoxypropanoic acid, 25c | 2-methyl-2...)
Affinity DataEC50:  4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28712(2-[4-({[2-(4-chlorophenyl)-4-methyl-1,3-thiazol-5-...)
Affinity DataEC50:  10nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28713(2-methyl-2-[4-({[4-methyl-2-(4-nitrophenyl)-1,3-th...)
Affinity DataEC50:  30nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28714(2-[4-({[2-(4-methoxyphenyl)-4-methyl-1,3-thiazol-5...)
Affinity DataEC50:  10nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28715(2-[4-({[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-...)
Affinity DataEC50:  40nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28716(2-methyl-2-(4-{[(4-methyl-2-phenyl-1,3-thiazol-5-y...)
Affinity DataEC50:  120nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28717(2-methyl-2-phenoxypropanoic acid, 25i | 2-methyl-2...)
Affinity DataEC50:  4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28718(2-methyl-2-phenoxypropanoic acid, 25j | 2-methyl-2...)
Affinity DataEC50:  465nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28719(2-[4-({[2-(4-aminophenyl)-4-methyl-1,3-thiazol-5-y...)
Affinity DataEC50:  5.64E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28720(2-methyl-2-phenoxypropanoic acid, 25l | 2-{4-[({2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28721(2-[4-({[2-(4-hydroxyphenyl)-4-methyl-1,3-thiazol-5...)
Affinity DataEC50: >1.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28722(2-methyl-2-phenoxypropanoic acid, 41 | 2-methyl-2-...)
Affinity DataEC50:  1.89E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28723(2-methyl-2-[4-({[4-(trifluoromethyl)-2-[4-(trifluo...)
Affinity DataEC50:  4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  1nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28702(2-[2-methyl-4-(2-{4-methyl-2-[4-(trifluoromethyl)p...)
Affinity DataEC50:  4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28703(2-methyl-2-[4-(2-{4-methyl-2-[4-(trifluoromethyl)p...)
Affinity DataEC50:  20nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28704(2-methyl-2-[4-({4-methyl-2-[4-(trifluoromethyl)phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28705(2-methyl-2-(4-{[({4-methyl-2-[4-(trifluoromethyl)p...)
Affinity DataEC50:  4.05E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  2.83E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28707(2-methyl-2-phenoxypropanoic acid, 27 | 2-methyl-2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28708(2-methyl-2-phenoxypropanoic acid, 34 | 2-methyl-2-...)
Affinity DataEC50:  6.26E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28709(2-methyl-2-phenoxypropanoic acid, 37 | 2-methyl-2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28710(2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazo...)
Affinity DataEC50: >1.00E+4nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28711(2-methyl-2-phenoxypropanoic acid, 25c | 2-methyl-2...)
Affinity DataEC50:  4.60E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28712(2-[4-({[2-(4-chlorophenyl)-4-methyl-1,3-thiazol-5-...)
Affinity DataEC50:  5.40E+3nMAssay Description:The ligand binding domain for PPAR was fused to the yeast transcription factor GAL4 DNA binding domain. CV-1 cells were transiently transfected with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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