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Found 33 with Last Name = 'siles' and Initial = 'r'
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352495(CHEMBL1824555)
Affinity DataKi:  880nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352496(CHEMBL1824556)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352497(CHEMBL1824553)
Affinity DataKi:  1.75E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352498(CHEMBL1824554)
Affinity DataKi:  1.97E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352499(CHEMBL1824551)
Affinity DataKi:  2.27E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352500(CHEMBL1824550)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352501(CHEMBL1824559)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352502(CHEMBL1824549)
Affinity DataKi:  5.43E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352503(CHEMBL1824552)
Affinity DataKi:  6.89E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352504(CHEMBL1824546)
Affinity DataKi:  8.91E+3nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352505(CHEMBL1824544)
Affinity DataKi:  1.37E+4nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352506(CHEMBL1824558)
Affinity DataKi:  3.92E+4nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50352507(CHEMBL1824542)
Affinity DataKi:  6.25E+4nMAssay Description:Inhibition of human thrombin using chromogenic Sar-Pro-Arg p-nitroanilide dihydrochloride as substrate pre-incubated for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189273(1-(7-bromo-3,4-dihydronaphthalen-1(2H)-ylidene)thi...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189279(1-(bis(3-bromophenyl)methylene)thiosemicarbazide |...)
Affinity DataIC50:  24nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189280(1-((3-bromophenyl)(phenyl)methylene)thiosemicarbaz...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189271(1-(6-bromo-2,3-dihydrochromen-4-ylidene)thiosemica...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189278(6-bromo-2,3-dihydro-4H-thiochromen-4-one thiosemic...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189263(1-(7-bromo-3,4-dihydronaphthalen-1-yl)prop-2-en-1-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189274(6,8-dibromo-2,3-dihydro-4H-thiochromen-4-one thios...)
Affinity DataIC50:  820nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189265(1-(1-(3-nitrophenyl)propylidene)thiosemicarbazide ...)
Affinity DataIC50:  860nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189261(1-(5-bromo-3,4-dihydronaphthalen-1(2H)-ylidene)thi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189272(1-(3,4-dihydronaphthalen-1-yl)ethanone | CHEMBL378...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189270(1-(2,3-dihydrothiochromen-4-ylidene)thiosemicarbaz...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189267(1-(1-(3-aminophenyl)propylidene)thiosemicarbazide ...)
Affinity DataIC50: >3.64E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189266(1-(3-(4-bromophenyl)cyclopentylidene)thiosemicarba...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189269(1-(3-(4-bromophenyl)cyclohexylidene)thiosemicarbaz...)
Affinity DataIC50: >7.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189262(1-(3,4-dihydrochromen-2-ylidene)thiosemicarbazide ...)
Affinity DataIC50: >1.60E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189264(1-(2,3-dihydrochromen-4-ylidene)thiosemicarbazide ...)
Affinity DataIC50: >1.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189268(1-(2,3-dihydroinden-1-ylidene)thiosemicarbazide | ...)
Affinity DataIC50: >1.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189276(1-(1-(3,4-dihydronaphthalen-1-yl)ethylidene)thiose...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189277(2,3-dihydro-4H-thiochromen-4-one thiosemicarbazone...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50189275(1-(1-(3-hydroxyphenyl)propylidene)thiosemicarbazid...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed