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Found 18 with Last Name = 'simoneaux' and Initial = 'r'
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175402(CHEMBL371435 | N-(2,4-difluorobenzyl)-N-((4-(4-cya...)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175406(CHEMBL200291 | N-((4-(4-cyanobenzyl)-4H-1,2,4-tria...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175395(CHEMBL199965 | N-(2,4-difluorobenzyl)-N-((4-(4-cya...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175407(CHEMBL371484 | N-(2,4-difluorobenzyl)-N-((4-(4-cya...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175392(CHEMBL371010 | N-((4-(4-cyanobenzyl)-4H-1,2,4-tria...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175408(CHEMBL371423 | N-(2,4-difluorobenzyl)-N-((4-((5-cy...)
Affinity DataIC50:  5.5nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175394(CHEMBL200193 | N-((4-(4-cyanobenzyl)-4H-1,2,4-tria...)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175400(CHEMBL201315 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  26nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175403(CHEMBL201299 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  28.3nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175401(CHEMBL199468 | N-((4-(4-cyanobenzyl)-4H-1,2,4-tria...)
Affinity DataIC50:  44nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175405(CHEMBL201066 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  53.2nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175397(CHEMBL370381 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  61nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175399(CHEMBL199365 | N-((4-(4-cyanobenzyl)-4H-1,2,4-tria...)
Affinity DataIC50:  75nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175393(CHEMBL200343 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  89.3nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175409(CHEMBL426837 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  96.5nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175398(CHEMBL381432 | N-(4-bromophenethyl)-N-((4-(4-cyano...)
Affinity DataIC50:  99.3nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175404(CHEMBL200829 | N-(2,4-difluorobenzyl)-N-((1-(4-cya...)
Affinity DataIC50:  187nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50175396(CHEMBL199491 | N-(2,4-difluorobenzyl)-N-((1-(4-cya...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against K-Ras farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed