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Found 5 with Last Name = 'simons' and Initial = 'ss'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50012202(17-(2-Bromo-acetyl)-9-fluoro-11,17-dihydroxy-10,13...)
Affinity DataIC50:  130nMAssay Description:Partial agonist(20%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50012201(9-Fluoro-11,17-dihydroxy-17-[2-(2-isothiocyanato-e...)
Affinity DataIC50:  440nMAssay Description:Partial agonist(48%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50012200(2,6-Bis-trifluoromethyl-benzoic acid 2-(9-fluoro-1...)
Affinity DataIC50:  770nMAssay Description:Antagonistic effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50012202(17-(2-Bromo-acetyl)-9-fluoro-11,17-dihydroxy-10,13...)
Affinity DataEC50:  8.30E+9nMAssay Description:Partial agonist (20%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50012201(9-Fluoro-11,17-dihydroxy-17-[2-(2-isothiocyanato-e...)
Affinity DataEC50:  9.10E+9nMAssay Description:Partial agonist (48%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed