Affinity DataIC50: 100nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair