TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Texas-Arlington
Curated by ChEMBL
University Of Texas-Arlington
Curated by ChEMBL
Affinity DataIC50: 7.97E+3nMAssay Description:Antagonist activity at human PPARgamma LBD expressed in yeast AH109 cells assessed as reduction in rosiglitazone-stimulated PPARgamma/CBP interaction...More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Birla Institute Of Technology
Curated by ChEMBL
Birla Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of c-erbB2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.37E+4nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair