TargetTransporter(Rattus norvegicus)
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-nisoxetine from NET in Sprague-Dawley rat brain prefrontal cortex incubated for 180 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus)
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-nisoxetine from NET in Sprague-Dawley rat brain prefrontal cortex incubated for 180 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-citalopram from SERT in Sprague-Dawley rat brainstem incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-WIN 3542875 from DAT in Sprague-Dawley rat brain striatum incubated for 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus)
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]-nisoxetine from NET in Sprague-Dawley rat brain prefrontal cortex incubated for 180 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus)
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [3H]-nisoxetine from NET in Sprague-Dawley rat brain prefrontal cortex incubated for 180 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 785nMAssay Description:Displacement of [3H]-citalopram from SERT in Sprague-Dawley rat brainstem incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 795nMAssay Description:Displacement of [3H]-citalopram from SERT in Sprague-Dawley rat brainstem incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 964nMAssay Description:Displacement of [3H]-WIN 3542875 from DAT in Sprague-Dawley rat brain striatum incubated for 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 1.14E+3nMAssay Description:Displacement of [3H]-citalopram from SERT in Sprague-Dawley rat brainstem incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 1.54E+3nMAssay Description:Displacement of [3H]-WIN 3542875 from DAT in Sprague-Dawley rat brain striatum incubated for 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 4.87E+3nMAssay Description:Displacement of [3H]-WIN 3542875 from DAT in Sprague-Dawley rat brain striatum incubated for 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus)
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxetine from NET in Sprague-Dawley rat brain prefrontal cortex incubated for 180 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-WIN 3542875 from DAT in Sprague-Dawley rat brain striatum incubated for 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-citalopram from SERT in Sprague-Dawley rat brainstem incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus)
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
National Institutes Of Drug Abuse - Intramural Research Program
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxetine from NET in Sprague-Dawley rat brain prefrontal cortex incubated for 180 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of rat GAT1 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.17E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of re-uptake of [3H]-dopamine at human DAT expressed in HEK293 cells preincubated for 5 mins followed by [3H]-dopamine addition measured a...More data for this Ligand-Target Pair