Compile Data Set for Download or QSAR
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Found 82 with Last Name = 'skeean' and Initial = 'r'
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012250(CHEMBL58947 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012246(CHEMBL58153 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012246(CHEMBL58153 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50282993((2S,4R)-4-Cyclohexyl-2-hydroxy-3-((R)-3-methylsulf...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012251(2-{2-(1-Cyclohexylmethyl-2,3-dihydroxy-5-methyl-he...)
Affinity DataIC50:  0.230nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012246(CHEMBL58153 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.280nMAssay Description:Inhibitory concentration against human reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035820(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37830)
Affinity DataIC50:  0.450nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012249(CHEMBL58256 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.680nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006202(3-Amino-N-[1-[1-(1-cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.75nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012257(CHEMBL299252 | N-[1-Cyclohexylmethyl-3,3-difluoro-...)
Affinity DataIC50:  0.790nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM17941((2S,4S,5S)-5-[(2S)-2-[(2S)-2-benzyl-3-[(2-methylpr...)
Affinity DataIC50:  0.830nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012252(CHEMBL57492 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012247(4-(1-Cyclohexylmethyl-2,3-dihydroxy-5-methyl-hexyl...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035832(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL35471)
Affinity DataIC50:  1.80nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035825(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL34554)
Affinity DataIC50:  3.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012255(CHEMBL293328 | N-[1-Cyclohexylmethyl-2-hydroxy-3-(...)
Affinity DataIC50:  4nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012253(CHEMBL56982 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50282993((2S,4R)-4-Cyclohexyl-2-hydroxy-3-((R)-3-methylsulf...)
Affinity DataIC50:  24nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012250(CHEMBL58947 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  27nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012254(CHEMBL60535 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  27nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012247(4-(1-Cyclohexylmethyl-2,3-dihydroxy-5-methyl-hexyl...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035829(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34853)
Affinity DataIC50:  30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012246(CHEMBL58153 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  36nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012246(CHEMBL58153 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  36nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]-etorphine as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012249(CHEMBL58256 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  43nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012246(CHEMBL58153 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  46nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035834(Ac-Trp-L-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL287753)
Affinity DataIC50:  50nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035833(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37984)
Affinity DataIC50:  70nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012253(CHEMBL56982 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012252(CHEMBL57492 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50: >100nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012256(CHEMBL431751 | N-{1-[1-Hydroxy-2-(2-morpholin-4-yl...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration against human reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035822(Ac-Trp-L-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL37983)
Affinity DataIC50:  300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012254(CHEMBL60535 | N-(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012257(CHEMBL299252 | N-[1-Cyclohexylmethyl-3,3-difluoro-...)
Affinity DataIC50:  515nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035823(Ac-Trp-D-Pro-Asp-Phe-NH2 | Ac-Trp-Pro-Asp-Phe-NH2 ...)
Affinity DataIC50:  600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035828(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37900)
Affinity DataIC50:  600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035821(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34916)
Affinity DataIC50:  800nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035833(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37984)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035823(Ac-Trp-D-Pro-Asp-Phe-NH2 | Ac-Trp-Pro-Asp-Phe-NH2 ...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035828(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37900)
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for binding affinity towards Cholecystokinin type A receptor by measuring its ability to displace [125I]-BH-CCK-8 from rat pancre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035825(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL34554)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035820(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37830)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012256(CHEMBL431751 | N-{1-[1-Hydroxy-2-(2-morpholin-4-yl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006202(3-Amino-N-[1-[1-(1-cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012255(CHEMBL293328 | N-[1-Cyclohexylmethyl-2-hydroxy-3-(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM17941((2S,4S,5S)-5-[(2S)-2-[(2S)-2-benzyl-3-[(2-methylpr...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035831(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL290444)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50225752(CHEMBL46012)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of Guinea Pig cAMP specific phosphodiesterase (PDE III)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035836((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035826((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  7.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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