Affinity DataIC50: 0.180nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Inhibitory concentration against human reninMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.830nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]-etorphine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against human reninMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
Affinity DataIC50: 515nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for binding affinity towards Cholecystokinin type A receptor by measuring its ability to displace [125I]-BH-CCK-8 from rat pancre...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Bovine Cathepsin D.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory concentration on Bovine Cathepsin DMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Guinea Pig cAMP specific phosphodiesterase (PDE III)More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair