Affinity DataKi: 16nMAssay Description:Binding affinity against Glutamate RacemaseMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 9.60nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 10.1nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 225nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
State University Of New York-Esf
Curated by ChEMBL
State University Of New York-Esf
Curated by ChEMBL
Affinity DataIC50: 695nMAssay Description:Inhibition of PI3 kinase p110alpha/p85alpha complexMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of Adenosine receptor A1More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Adenosine receptor A1More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Adenosine receptor A1More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Adenosine receptor A1More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 95nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 102nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 103nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 411nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 474nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 633nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 833nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 1.44E+3nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 193nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 269nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 328nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 352nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: >4.00E+3nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: >4.00E+3nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 366nMAssay Description:Agonist activity at Toll-like receptor 7More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at TLR7 in human PBMC assessed as induction of type 1 interferon productionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at TLR7 in human PBMC assessed as induction of type 1 interferon productionMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Agonist activity at TLR7 in human PBMC assessed as induction of type 1 interferon productionMore data for this Ligand-Target Pair
Affinity DataEC50: 26.9nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 28.6nMAssay Description:Agonist activity at TLR7 in human PBMC assessed as induction of type 1 interferon productionMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 32.1nMAssay Description:Agonist activity at TLR7More data for this Ligand-Target Pair
Affinity DataEC50: 45.8nMAssay Description:Agonist activity at TLR7 in human PBMC assessed as induction of type 1 interferon productionMore data for this Ligand-Target Pair