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Found 17 with Last Name = 'smith' and Initial = 'rm'
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297503(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297505(CHEMBL563988 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297506(CHEMBL551074 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297505(CHEMBL563988 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297504(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50001709(4-cyclopropylmethyl-(13R)-12-oxa-4-azapentacyclo[9...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297505(CHEMBL563988 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297506(CHEMBL551074 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50001709(4-cyclopropylmethyl-(13R)-12-oxa-4-azapentacyclo[9...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297503(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297504(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297503(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297506(CHEMBL551074 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50001709(4-cyclopropylmethyl-(13R)-12-oxa-4-azapentacyclo[9...)
Affinity DataKi:  213nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297504(17-(cyclopropylmethyl)-3,14-dihydroxy-6beta-(N,N-d...)
Affinity DataKi:  334nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50537996(CHEMBL4632827)
Affinity DataKd:  550nMAssay Description:Binding affinity to wild-type human partial length JAK1 JH2 pseudokinase domain (R537 to D855 residues) expressed in mammalian expression system at 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50537996(CHEMBL4632827)
Affinity DataKd:  410nMAssay Description:Binding affinity to wild-type human partial length PIK3C3 (S282 to H879 residues) expressed in mammalian expression system at 10 uM by Kinomescan met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed