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Found 23 with Last Name = 'smith' and Initial = 'wj'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055721(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity was determined in vitro on rat striatum using [3H]-N-propylnorapomorphine against Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055719(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  8.60nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055725(3-{4-[2-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-eth...)
Affinity DataKi:  8.70nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50002173(3-(4-(3,6-dihydro-4-phenyl-1(2H)-pyridinyl)butyl)-...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055731(3-{4-[2-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-eth...)
Affinity DataKi:  28nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055721(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  29nMAssay Description:In vitro binding affinity of the compound towards human recombinant Dopamine receptor D3 receptor expressed in CHO-K1 cells was determined using [3H]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055727(5-Methoxy-3-{4-[2-(4-pyridin-2-yl-piperazin-1-yl)-...)
Affinity DataKi:  29nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055721(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  50nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055721(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  73nMAssay Description:In vitro binding affinity of the compound towards human recombinant Dopamine receptor D4 expressed in CHO-K1 cells was determined using [3H]-spiperon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055728(1-Methyl-3-{4-[2-(4-pyridin-2-yl-piperazin-1-yl)-e...)
Affinity DataKi:  83nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055723(3-[4-(4-Pyridin-2-yl-piperazin-1-ylmethyl)-cyclohe...)
Affinity DataKi:  85nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055734(5-Fluoro-3-{4-[2-(4-pyridin-2-yl-piperazin-1-yl)-e...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055720(3-[4-(4-Pyridin-2-yl-piperazin-1-ylmethyl)-cyclohe...)
Affinity DataKi:  122nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055729(3-{4-[2-(4-Phenyl-piperazin-1-yl)-ethyl]-cyclohexy...)
Affinity DataKi:  124nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055733(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  139nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055722(3-{4-[2-(4-Pyrimidin-2-yl-piperazin-1-yl)-ethyl]-c...)
Affinity DataKi:  161nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055735(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataKi:  270nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055724(1-[2-((S)-4-Phenyl-cyclohex-3-enyl)-ethyl]-4-pyrid...)
Affinity DataKi:  412nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055726(3-[4-(4-Pyridin-2-yl-piperazin-1-yl)-cyclohexyl]-1...)
Affinity DataKi:  457nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055730(3-{4-[2-(4-Thiophen-2-yl-3,6-dihydro-2H-pyridin-1-...)
Affinity DataKi:  630nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055732(3-(4-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethyl...)
Affinity DataKi:  645nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055718(3-[4-(4-Pyridin-2-yl-piperazin-1-yl)-cyclohexyl]-1...)
Affinity DataKi:  2.60E+3nMAssay Description:In vitro binding affinity for dopamine receptor D2 on rat striatal membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Division Of Warner Lambert

Curated by ChEMBL
LigandPNGBDBM50055721(3-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataEC50:  2.80nMAssay Description:Inhibition of [3H]-thymidine uptake by Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed