TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]-dexamethasone binding to human Glucocorticoid ReceptorMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Affinity for human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of [3H]-dexamethasone binding to human Glucocorticoid ReceptorMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of [3H]-dexamethasone binding to human Glucocorticoid ReceptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Affinity for human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 146nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 172nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 194nMAssay Description:Inhibition of [3H]-dexamethasone binding to human Glucocorticoid ReceptorMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 252nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 289nMAssay Description:Affinity for human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 312nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 357nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Affinity for human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 442nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration against mammalian Squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory activity against Squalene synthase from ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 505nMAssay Description:In vitro for inhibitory activity against Squalene synthase in ratMore data for this Ligand-Target Pair