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Found 35 with Last Name = 'sobarzo-sánchez' and Initial = 'e'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358012(CHEMBL1651055)
Affinity DataIC50:  0.830nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202337((S)-3-iodo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358015(CHEMBL1917530)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358009(CHEMBL1651054)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358014(CHEMBL1917529)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358010(CHEMBL1917527)
Affinity DataIC50:  44nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202340((S)-3-bromo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetra...)
Affinity DataIC50:  66nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50269193(3-Chloroboldine | CHEMBL524439)
Affinity DataIC50:  81nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202337((S)-3-iodo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50:  96nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50209211(3,8-dibromoboldine | CHEMBL388564)
Affinity DataIC50:  206nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202318((+)-boldine | (S)-(+)-Boldine | (S)-1,10-dimethoxy...)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202318((+)-boldine | (S)-(+)-Boldine | (S)-1,10-dimethoxy...)
Affinity DataIC50:  520nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358011(CHEMBL461133)
Affinity DataIC50:  720nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50269193(3-Chloroboldine | CHEMBL524439)
Affinity DataIC50:  720nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50202340((S)-3-bromo-1,10-dimethoxy-6-methyl-5,6,6a,7-tetra...)
Affinity DataIC50:  1.05E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358013(CHEMBL1917528)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50209211(3,8-dibromoboldine | CHEMBL388564)
Affinity DataIC50:  1.91E+3nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358016(CHEMBL1917531)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  6.56E+3nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  7.54E+3nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358017(CHEMBL1917532)
Affinity DataIC50:  9.81E+3nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358008(CHEMBL1917526)
Affinity DataIC50:  2.73E+4nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358017(CHEMBL1917532)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358016(CHEMBL1917531)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  6.34E+4nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358011(CHEMBL461133)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358012(CHEMBL1651055)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358013(CHEMBL1917528)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358014(CHEMBL1917529)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358010(CHEMBL1917527)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358009(CHEMBL1651054)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358008(CHEMBL1917526)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50358015(CHEMBL1917530)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataIC50:  3.61E+5nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed