TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.56nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human influenza A virus A/Aichi/2/1968(H3N2) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.66nMAssay Description:Inhibition of human influenza A virus A/Aichi/2/1968(H3N2) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Inhibition of CDC25B in presence of 2 mM DTTMore data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of CDC25A in presence of 2 mM DTTMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: >1.29E+3nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: >1.42E+3nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: >1.48E+3nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair
TargetIsoleucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Riken (Institute Of Physical And Chemical Research)
Curated by ChEMBL
Affinity DataIC50: >1.51E+3nMAssay Description:Inhibition of IleRSMore data for this Ligand-Target Pair