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Found 132 with Last Name = 'solomon' and Initial = 'vr'
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50143115(3-Phenyl-6-(pyridin-2-ylmethoxy)-[1,2,4]triazolo[3...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity to recombinant human GABA-A alpha5beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50143115(3-Phenyl-6-(pyridin-2-ylmethoxy)-[1,2,4]triazolo[3...)
Affinity DataKi:  0.710nMAssay Description:Binding affinity to recombinant human GABA-A alpha3beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50162235(6-phenyl-4,5,7,8-tetraazatetracyclo[9.2.2.02,10.03...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to recombinant human GABA-A alpha5beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50156083(3-tert-Butyl-7-(5-methyl-isoxazol-3-yl)-2-(2-methy...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant human GABA-A alpha5beta3gamma2 receptor expressed in mouse L(tk-) cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50143115(3-Phenyl-6-(pyridin-2-ylmethoxy)-[1,2,4]triazolo[3...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to recombinant human GABA-A alpha1beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50156083(3-tert-Butyl-7-(5-methyl-isoxazol-3-yl)-2-(2-methy...)
Affinity DataKi:  3nMAssay Description:Inverse agonist activity at recombinant human GABA-A alpha5beta3gamma2 receptor expressed in mouse L(tk-) cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50162235(6-phenyl-4,5,7,8-tetraazatetracyclo[9.2.2.02,10.03...)
Affinity DataKi:  12nMAssay Description:Binding affinity to recombinant human GABA-A alpha3beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50143106(6-Benzyloxy-3-phenyl-[1,2,4]triazolo[3,4-a]phthala...)
Affinity DataKi:  38nMAssay Description:Binding affinity to recombinant human GABA-A alpha5beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50143106(6-Benzyloxy-3-phenyl-[1,2,4]triazolo[3,4-a]phthala...)
Affinity DataKi:  41nMAssay Description:Binding affinity to recombinant human GABA-A alpha3beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50162235(6-phenyl-4,5,7,8-tetraazatetracyclo[9.2.2.02,10.03...)
Affinity DataKi:  71nMAssay Description:Binding affinity to recombinant human GABA-A alpha1beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50143106(6-Benzyloxy-3-phenyl-[1,2,4]triazolo[3,4-a]phthala...)
Affinity DataKi:  280nMAssay Description:Binding affinity to recombinant human GABA-A alpha1beta3gamma2 receptor expressed in L(tk) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282700(CHEMBL35324 | N-(2-Chloro-benzyl)-N-{2-methyl-4-ox...)
Affinity DataIC50:  0.0600nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282704(CHEMBL285433 | N-(2-Chloro-benzyl)-N-{2-ethyl-4-ox...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282705(CHEMBL290669 | N-Benzyl-N-{2-isopropyl-4-oxo-3-[2'...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282708(CHEMBL289472 | Thiophene-2-carboxylic acid benzyl-...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282710(CHEMBL34082 | N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282703(CHEMBL35638 | N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282701(CHEMBL285432 | N-Benzyl-N-{2-methyl-4-oxo-3-[2'-(1...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282702(CHEMBL290768 | Thiophene-2-carboxylic acid benzyl-...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50282706(CHEMBL276853 | N-{2-Ethyl-4-oxo-3-[2'-(1H-tetrazol...)
Affinity DataIC50:  0.460nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50615602(CHEMBL5278845)
Affinity DataIC50:  0.460nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50615601(CHEMBL302102 | L-159689)
Affinity DataIC50:  1nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615600(CHEMBL5273148)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615596(CHEMBL5286548)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615595(CHEMBL5268759)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615594(CHEMBL5288172)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615593(CHEMBL5287291)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615592(CHEMBL5283610)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615597(CHEMBL5282201)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615599(CHEMBL5271165)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615598(CHEMBL5266971)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615583(CHEMBL321678)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615584(CHEMBL5267424)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615585(CHEMBL111859)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615586(CHEMBL113019)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615587(CHEMBL109881)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615588(CHEMBL320036)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615589(CHEMBL264198)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615590(CHEMBL5289121)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615591(CHEMBL5289689)
Affinity DataIC50:  3nMAssay Description:Inhibition of human TSMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensinogen(Homo sapiens)TBA
LigandPNGBDBM50282821(2-Butyl-6-((2S,3aR)-2-methyl-hexahydro-pyrrolo[1,2...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of angiotensin II (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50213087(CHEMBL14748)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50213198(CHEMBL15225)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50213086(CL-329167)
Affinity DataIC50:  18nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50213084(CHEMBL15118)
Affinity DataIC50:  18nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50213196(CHEMBL15154)
Affinity DataIC50:  18nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAngiotensinogen(Homo sapiens)TBA
LigandPNGBDBM50615610(CHEMBL5275762)
Affinity DataIC50:  22nMAssay Description:Inhibition of angiotensin II (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensinogen(Homo sapiens)TBA
LigandPNGBDBM50615611(CHEMBL5281619)
Affinity DataIC50:  22nMAssay Description:Inhibition of angiotensin II (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensinogen(Homo sapiens)TBA
LigandPNGBDBM50615609(CHEMBL295174)
Affinity DataIC50:  27nMAssay Description:Inhibition of angiotensin II (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAngiotensinogen(RAT)TBA
LigandPNGBDBM50615607(CHEMBL415982)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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