Affinity DataKi: 10nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 1.37E+4nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 2.13E+5nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+5nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+5nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+6nMAssay Description:Inhibition of tissue kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+6nMAssay Description:Inhibition of tissue kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+6nMAssay Description:Inhibition of plasma kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+6nMAssay Description:Inhibition of plasma kallikreinMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human ERG channel IKr expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human ERG channel IKr expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human ERG channel IKr expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of recombinant human ERG channel IKr expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of recombinant CYP2C9 (unknown origin) after 10 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.71E+3nMAssay Description:Inhibition of recombinant CYP3A4 (unknown origin) after 3 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant CYP1A2 (unknown origin) after 10 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant CYP2D6 (unknown origin) after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of recombinant human ERG channel IKr expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant human ERG channel IKr expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair