Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13.7nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Modulation of mGluR5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 24.9nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26.7nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30.5nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30.8nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31.2nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33.8nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33.9nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33.9nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 36.7nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38.5nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38.9nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 42.2nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 42.7nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 44.8nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45.3nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45.3nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 47.7nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48.9nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50.4nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50.6nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50.7nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52.6nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 53.4nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54.1nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 56.4nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 56.9nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 57.4nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 57.6nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64.6nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 65.4nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 67.7nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of peptidase activity of human recombinant LTA4H expressed in Escherichia coli BL21-AI/pRAREMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of hydrolase activity of human recombinant LTA4H expressed in Escherichia coli BL21-AI/pRARE assessed as LTB4 formation by tandem quadrupo...More data for this Ligand-Target Pair
Affinity DataIC50: 74.4nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 76.2nMAssay Description:Inhibition of recombinant human DPP4 after 1 hr by fluorescence assayMore data for this Ligand-Target Pair