Affinity DataKi: 0.00400nM ΔG°: -66.1kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
Affinity DataKi: 0.0110nM ΔG°: -63.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
Affinity DataKi: 0.0120nM ΔG°: -63.4kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
Affinity DataKi: 0.112nM ΔG°: -57.7kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.430nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.320nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.200nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 30nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 2.40nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M4 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.356nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M4 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 6.80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 41nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.383nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Oak Ridge National Laboratory (Ornl)
Curated by ChEMBL
Affinity DataKd: 0.230nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair