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Found 78 with Last Name = 'soulère' and Initial = 'l'
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089703(CHEMBL29507 | N-[4-(3-Nitrooxy-propyl)-phenyl]-[1,...)
Affinity DataKi:  200nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089708(2-(acetylamino)-N-{4-[(4,6-diamino-1,3,5-triazin-2...)
Affinity DataKi:  580nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089698(2-(acetylamino)-N-[2-(6-amino-9H-purin-9-yl)ethyl]...)
Affinity DataKi:  620nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089705(9-(2-Nitrooxy-ethyl)-9H-purin-6-ylamine | CHEMBL26...)
Affinity DataKi:  1.90E+3nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366636(CHEMBL605462)
Affinity DataKi:  3.47E+3nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM108256(CHEMBL2205239 | US8609833, 87)
Affinity DataKi:  1.23E+4nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50421414(CYMELARSEN | Cymelarsan)
Affinity DataKi:  2.29E+4nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089701(5,7-Diamino-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ol...)
Affinity DataKi:  1.17E+5nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089706(2-(acetylamino)-N-(6-aminopyridin-3-yl)-3-methyl-3...)
Affinity DataKi:  4.04E+5nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089704(CHEMBL25961 | nitrooxymethyl-benzene)
Affinity DataKi: >1.00E+6nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366635(CHEMBL73188)
Affinity DataKi: >1.00E+6nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350660(CHEMBL1813552)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373056(CHEMBL261163)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350661(CHEMBL1813553)
Affinity DataIC50:  2.70E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373048(CHEMBL184106)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350666(CHEMBL1813558)
Affinity DataIC50:  3.40E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373057(CHEMBL261162)
Affinity DataIC50:  3.60E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350659(CHEMBL1813551)
Affinity DataIC50:  4.00E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350669(CHEMBL1813546)
Affinity DataIC50:  4.90E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373055(CHEMBL408369)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373047(CHEMBL260235)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350649(CHEMBL1813536)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350670(CHEMBL1813559)
Affinity DataIC50:  5.30E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350653(CHEMBL1813540)
Affinity DataIC50:  5.80E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350648(CHEMBL1813535)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350654(CHEMBL1813541)
Affinity DataIC50:  6.20E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373052(CHEMBL404926)
Affinity DataIC50:  6.40E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350657(CHEMBL1813547)
Affinity DataIC50:  6.50E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262515(CHEMBL453930 | N-(4-bromo-2-oxo-2,5-dihydrofuran-3...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50262517(CHEMBL448263 | N-(4-chloro-2-oxo-2,5-dihydrofuran-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of LuxR-dependent Vibrio fischeri quorum sensing assessed as reduction in 3-oxo-hexanoyihomoserine-induced bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50323389(CHEMBL1208858 | Calmidazolium)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of LuxR-dependent quorum sensing in Vibrio fischeri assessed as reduction of 3-oxo-C6-HSL-induced bioluminescence intensityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373054(CHEMBL408296)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350650(CHEMBL1813537)
Affinity DataIC50:  7.30E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373053(CHEMBL260905)
Affinity DataIC50:  7.80E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350668(CHEMBL1813545)
Affinity DataIC50:  8.90E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373050(CHEMBL258584)
Affinity DataIC50:  9.40E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350652(CHEMBL1813539)
Affinity DataIC50:  9.80E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350665(CHEMBL1813557)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373049(CHEMBL408121)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373051(CHEMBL404924)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350662(CHEMBL1813554)
Affinity DataIC50:  1.47E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350647(CHEMBL1813534)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50028094((1S,4S)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-te...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of LuxR-dependent quorum sensing in Vibrio fischeri assessed as reduction of 3-oxo-C6-HSL-induced bioluminescence intensityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350664(CHEMBL1813556)
Affinity DataIC50:  3.30E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50356098(CHEMBL1911953)
Affinity DataIC50:  3.40E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 containing Photorhabdus luminescens LuxCDABE assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50350658(CHEMBL1813550)
Affinity DataIC50:  3.50E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50356106(CHEMBL1911959)
Affinity DataIC50:  4.00E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 containing Photorhabdus luminescens LuxCDABE assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of LuxR-dependent quorum sensing in Vibrio fischeri assessed as reduction of 3-oxo-C6-HSL-induced bioluminescence intensityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50389272(CHEMBL2063565)
Affinity DataIC50:  5.10E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 coexpressing LuxCDABE assessed as inhibition of 3-oxoC6-HSL-induced q...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50356104(CHEMBL1911955)
Affinity DataIC50:  5.20E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR expressed in Escherichia coli NM522 containing Photorhabdus luminescens LuxCDABE assessed as inhibition o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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