Compile Data Set for Download or QSAR
maximum 50k data
Found 195 with Last Name = 'spallarossa' and Initial = 'a'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354137(CHEMBL1836187)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]-WIN 55,212-2 from human CB2 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354135(CHEMBL1836189)
Affinity DataKi:  10.2nMAssay Description:Displacement of [3H]-WIN 55,212-2 from human CB2 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50354135(CHEMBL1836189)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]-CP-55,940 from human CB1 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247204(CHEMBL474125 | N-Cyclopropyl-1-(2,4-dichlorophenyl...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant PDE4D3 expressed in baculovirus system by radiometric assayMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  490nMAssay Description:Inhibition of human recombinant PDE4D1 expressed in baculovirus system by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224371(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(e...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142887(1-(tert-butyl)-3-(4-chlorophenyl)-4-aminopyrazolo[...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224368(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(m...)
Affinity DataKi:  600nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142880(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenet...)
Affinity DataKi:  700nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247415(5-(4-Chlorophenyl)-N-cyclopropyl-1-(2,4-dichloroph...)
Affinity DataKi:  850nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  930nMAssay Description:Inhibition of human recombinant PDE4D2 expressed in baculovirus system by radiometric assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247428(5-(4-Bromophenyl)-N-cyclopropyl-1-(2,4-dichlorophe...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247429(5-(4-Bromophenyl)-N-cycloheptyl-1-(2,4-dichlorophe...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247205(CHEMBL516381 | N-Cycloheptyl-1-(2,4-dichlorophenyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224376(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(p...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224385(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247430(1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-N-piperidi...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354134(CHEMBL1836188)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]-WIN 55,212-2 from human CB2 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224381(1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(m...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50299568(3-(Cyclopentyloxy)-4-methoxybenzaldehyde O-[3-(2,6...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of human recombinant PDE4D3 expressed in baculovirus system by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354136(CHEMBL1836121)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-WIN 55,212-2 from human CB2 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224388(CHEMBL238561 | N-(3-bromophenyl)-1-(2-chloro-2-phe...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50247430(1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-N-piperidi...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247416(5-(4-Bromophenyl)-1-(2,4-dichlorophenyl)-N-(4-meth...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224383(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224374(CHEMBL241749 | N-benzyl-1-(2-chloro-2-(4-chlorophe...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224387(1-(2-chloro-2-phenylethyl)-N-(2-chlorobenzyl)-6-(m...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142885(Benzyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfan...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224366(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-1H-p...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50299568(3-(Cyclopentyloxy)-4-methoxybenzaldehyde O-[3-(2,6...)
Affinity DataKi:  3.86E+3nMAssay Description:Inhibition of human recombinant PDE4D1 expressed in baculovirus system by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224386(CHEMBL399813 | N-(4-methoxyphenethyl)-1-(2-chloro-...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224367(1-(2-chloro-2-phenylethyl)-N-(2-chlorophenethyl)-6...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224382(CHEMBL399627 | N-(3-bromophenyl)-1-(2-chloro-2-(4-...)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224372(1-(2-chloro-2-phenylethyl)-N-(4-fluorobenzyl)-6-(m...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224384(1-(2-chloro-2-phenylethyl)-N-(3-fluorobenzyl)-6-(m...)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224380(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenethyl)-6...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224369(1-(2-chloro-2-phenylethyl)-6-(ethylthio)-N-pheneth...)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50299568(3-(Cyclopentyloxy)-4-methoxybenzaldehyde O-[3-(2,6...)
Affinity DataKi:  9.18E+3nMAssay Description:Inhibition of human recombinant PDE4D2 expressed in baculovirus system by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50354134(CHEMBL1836188)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP-55,940 from human CB1 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50354136(CHEMBL1836121)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP-55,940 from human CB1 receptor expressed in human HEK293 cells after 90 mins by radioligand assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224373(1-(2-chloro-2-phenylethyl)-N-(3-fluorophenethyl)-6...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224379(1-(2-chloro-2-phenylethyl)-N-(4-methylphenethyl)-6...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247390(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(4-met...)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224377(1-(2-chloro-2-phenylethyl)-N-(2-fluorobenzyl)-6-(m...)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50247415(5-(4-Chlorophenyl)-N-cyclopropyl-1-(2,4-dichloroph...)
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224378(CHEMBL239192 | N-(4-chlorobenzyl)-1-(2-chloro-2-ph...)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224375(CHEMBL401038 | N-(4-chlorophenethyl)-7-(2-chloro-2...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 195 total ) | Next | Last >>
Jump to: