Affinity DataKi: 1nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
Affinity DataKi: 727nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataKi: 765nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human plasma AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human erythrocytes AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human erythrocytes AChEMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche - Università
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Displacement of [3H]-pirenzepine binding to muscarinic M1 receptor in brain cortex of rat.More data for this Ligand-Target Pair