TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of [3H]-MPEP from human mGluR5More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.37E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5More data for this Ligand-Target Pair
Affinity DataIC50: 0.0820nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.670nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of BACE1 by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 151nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Displacement of [125I]U69593 from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 181nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of BACE1 by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 211nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 245nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 351nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of BACE1 by FRET assayMore data for this Ligand-Target Pair