BindingDB PrimarySearch

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM12372(1-{[5-(5-chlorothiophen-2-yl)-1,2-oxazol-3-yl]meth...)

Ki: 3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

MMDB PC cid PC sid PDB Patents Similars

Details PubMed MMDB
PDB

3D Structure (crystal)

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM12400(1-[(4-Chloro-phenylcarbamoyl)-methyl]-1H-indole-2-...)

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

DrugBank MMDB PC cid PC sid PDB Patents Similars

Details PubMed MMDB
PDB

3D Structure (crystal)

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590072(CHEMBL3904655)

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590086(CHEMBL5192536)

Ki: 4nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590082(CHEMBL5175184)

Ki: 6nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590073(CHEMBL5175600)

Ki: 7nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590087(CHEMBL5179837)

Ki: 8nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590097(CHEMBL5187449)

Ki: 9nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590083(CHEMBL5192808)

Ki: 11nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590078(CHEMBL5175799)

Ki: 12nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590081(CHEMBL5180386)

Ki: 13nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590099(CHEMBL5193338)

Ki: 37nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8117(Hydroxyethylene Sulfone 17b | N-[(2S,3R,5S)-1-(3-b...)

Ki: 45nM ΔG°: -41.9kJ/mole IC50: 85nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

MMDB PC cid PC sid PDB Similars

Details Article PubMed PDB

3D Structure (crystal)

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590075(CHEMBL5190215)

Ki: 49nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590084(CHEMBL5208176)

Ki: 51nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590089(CHEMBL5181980)

Ki: 52nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590080(CHEMBL5185736)

Ki: 55nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590074(CHEMBL5187415)

Ki: 56nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590088(CHEMBL5192209)

Ki: 57nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590071(CHEMBL5178354)

Ki: 63nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590096(CHEMBL5173515)

Ki: 65nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590077(CHEMBL5188689)

Ki: 70nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590076(CHEMBL5204725)

Ki: 162nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590079(CHEMBL5193560)

Ki: 188nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590070(CHEMBL5206688)

Ki: 204nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590093(CHEMBL5186260)

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590095(CHEMBL5199539)

Ki: 241nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8123(Hydroxyethylene Sulfone 18a | N-((1S,2R,4S)-1-(3-b...)

Ki: 370nM ΔG°: -36.7kJ/mole IC50: 530nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8124(Hydroxyethylene Sulfone 18b | N-((1S,2R,4S)-1-(3-b...)

Ki: 540nM ΔG°: -35.8kJ/mole IC50: 790nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590098(CHEMBL5194849)

Ki: 1.24E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8118(Hydroxyethylene Sulfone 17b- | N-[(2R,3S,5R)-1-(3-...)

Ki: 1.40E+3nM ΔG°: -33.4kJ/mole IC50: 2.00E+3nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590092(CHEMBL5205467)

Ki: 1.74E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8121((2R)-N-[(2S,3R,5S)-1-(3-bromophenyl)-7-(2,4-dichlo...)

Ki: 2.90E+3nM ΔG°: -31.6kJ/mole IC50: 4.20E+3nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590091(CHEMBL5202796)

Ki: 2.93E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8120(2-bromo-N-[(2S,3R,5S)-1-(3-bromophenyl)-7-(2,4-dic...)

Ki: 3.10E+3nM ΔG°: -31.4kJ/mole IC50: 4.50E+3nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590090(CHEMBL5175878)

Ki: 5.13E+3nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8119(Hydroxyethylene Sulfone 17c | N-[(2S,3R,5S)-1-(3-b...)

Ki: 7.00E+3nM ΔG°: -29.4kJ/mole IC50: 1.00E+4nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590100(CHEMBL5176283)

Ki: 1.48E+4nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Coagulation factor X(Homo sapiens (Human))
Leibniz-Forschungsinstitut F�R Molekulare Pharmakologie

Curated by ChEMBL

BDBM50590094(CHEMBL5205339)

Ki: 2.05E+4nMAssay Description:Inhibition of human fXa assessed as inhibition constant using Cbz-D-Arg-Gly-L-Arg-pNA as substrate preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8122((2R)-N-[(2R,3S,5R)-1-(3-bromophenyl)-7-(2,4-dichlo...)

Ki: >4.00E+4nM ΔG°: >-25.1kJ/mole IC50: >4.00E+4nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair

Dimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

BDBM8116(Hydroxyethylene Sulfone 17a | N-[(2S,3R,5S)-1-(3-b...)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM445676(Ex. 14/KM-06-64/(I-14) | US10683309, Example 14 | ...)

IC50: 11nMAssay Description:The full-length coding sequences of human TPH1 and TPH2 were PCR amplified, ligated into a MBP fusion vector (pMalc2x, New England Biolabs, MA, USA) ...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM445676(Ex. 14/KM-06-64/(I-14) | US10683309, Example 14 | ...)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM357735(KM-05-193/(I-209) | US10214530, Example 27)

IC50: 14nMAssay Description:Inhibition of N-terminal MBP-tagged full length human TPH2 assessed as reduction in 5-HTP formation incubated for 5 to 10 mins by fluorescence microp...More data for this Ligand-Target Pair

PC cid PC sid PDB

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM357737(KM-05-166/(I-206) | US10214530, Example 24)

IC50: 14nMAssay Description:These compounds according to the afore-mentioned examples were tested for tryptophan hydroxylase (TPH) inhibitory activity in a fluorescence-based in...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM357737(KM-05-166/(I-206) | US10214530, Example 24)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM357735(KM-05-193/(I-209) | US10214530, Example 27)

PC cid PC sid PDB

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM445677(Ex. 15/KM-06-96/(I-15) | US10683309, Example 15 | ...)

IC50: 14nMAssay Description:The full-length coding sequences of human TPH1 and TPH2 were PCR amplified, ligated into a MBP fusion vector (pMalc2x, New England Biolabs, MA, USA) ...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Tryptophan 5-hydroxylase 2(Homo sapiens (Human))
Max-DelbrÜCk-Centrum FÜR Molekulare Medizin

US Patent

BDBM445677(Ex. 15/KM-06-96/(I-15) | US10683309, Example 15 | ...)