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Found 42 with Last Name = 'spencer' and Initial = 'ja'
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50115622(2-Pyridazin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene | C...)
Affinity DataKi:  68.4nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50110260(2-Pyridin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene | 2-P...)
Affinity DataKi:  89nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  101nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50110259(2-Pyrimidin-5-yl-9-aza-bicyclo[4.2.1]non-2-ene | C...)
Affinity DataKi:  1.71E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50110258((6S)-2-(6-chloropyridin-3-yl)-9-azabicyclo[4.2.1]n...)
Affinity DataKi:  2.76E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50110263(2-Pyrazin-2-yl-9-aza-bicyclo[4.2.1]non-2-ene | CHE...)
Affinity DataKi:  5.77E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50115624(2-Pyridin-2-yl-9-aza-bicyclo[4.2.1]non-2-ene | CHE...)
Affinity DataKi:  4.75E+4nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50115623(2-Pyridin-4-yl-9-aza-bicyclo[4.2.1]non-2-ene | CHE...)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543044(CHEMBL4636926)
Affinity DataIC50:  16nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543037(CHEMBL4638471)
Affinity DataIC50:  20nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543029(CHEMBL4632789)
Affinity DataIC50:  40nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543033(CHEMBL4646806)
Affinity DataIC50:  50nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543047(CHEMBL4647878)
Affinity DataIC50:  63nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543049(CHEMBL4640045)
Affinity DataIC50:  79nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543043(CHEMBL4633472)
Affinity DataIC50:  100nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543038(CHEMBL4649257)
Affinity DataIC50:  126nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543045(CHEMBL4647230)
Affinity DataIC50:  158nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543046(CHEMBL4632438)
Affinity DataIC50:  251nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543037(CHEMBL4638471)
Affinity DataIC50:  316nMAssay Description:Inhibition of PI3Kdelta in whole blood (unknown origin) assessed as reduction in cytostim-induced IFNgamma productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543041(CHEMBL4646959)
Affinity DataIC50:  398nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543050(CHEMBL4649799)
Affinity DataIC50:  501nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543032(CHEMBL4645570)
Affinity DataIC50:  631nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543039(CHEMBL4637133)
Affinity DataIC50:  631nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543048(CHEMBL4641762)
Affinity DataIC50:  631nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543027(CHEMBL4644887)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543037(CHEMBL4638471)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543040(CHEMBL4640147)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543030(CHEMBL4645872)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543031(CHEMBL4636609)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543032(CHEMBL4645570)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of PI3Kdelta in whole blood (unknown origin) assessed as reduction in cytostim-induced IFNgamma productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543037(CHEMBL4638471)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543037(CHEMBL4638471)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543028(CHEMBL4646294)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543034(CHEMBL4634067)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543042(CHEMBL4632521)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543032(CHEMBL4645570)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543035(CHEMBL4649680)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543032(CHEMBL4645570)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543036(CHEMBL4633464)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543032(CHEMBL4645570)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543037(CHEMBL4638471)
Affinity DataKd:  4nMAssay Description:Binding affinity to PI3Kdelta (unknown origin) by SPR based van't Hoff analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50543032(CHEMBL4645570)
Affinity DataKd:  251nMAssay Description:Binding affinity to PI3Kdelta (unknown origin) by SPR based van't Hoff analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB