TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 68.4nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 101nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 2.76E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 5.77E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: 4.75E+4nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of PI3Kdelta in whole blood (unknown origin) assessed as reduction in cytostim-induced IFNgamma productionMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 398nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 501nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of PI3Kdelta in whole blood (unknown origin) assessed as reduction in cytostim-induced IFNgamma productionMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataKd: 4nMAssay Description:Binding affinity to PI3Kdelta (unknown origin) by SPR based van't Hoff analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gsk Medicines Research Centre
Curated by ChEMBL
Gsk Medicines Research Centre
Curated by ChEMBL
Affinity DataKd: 251nMAssay Description:Binding affinity to PI3Kdelta (unknown origin) by SPR based van't Hoff analysisMore data for this Ligand-Target Pair