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Found 30 with Last Name = 'spino' and Initial = 'm'
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional

Curated by ChEMBL
LigandPNGBDBM50127979(3-(2,5-Dioxo-pyrrolidin-1-yl)-benzoic acid | CHEMB...)
Affinity DataIC50:  33nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional

Curated by ChEMBL
LigandPNGBDBM50127981(3-(3-Carboxy-propionylamino)-benzoic acid | CHEMBL...)
Affinity DataIC50:  93nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164216(CHEMBL190022 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164222(CHEMBL193212 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50172756(Benzyl-methyl-prop-2-ynyl-amine | CHEMBL673 | Euto...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional

Curated by ChEMBL
LigandPNGBDBM50127978(3-(2,5-Dioxo-2,5-dihydro-pyrrol-1-yl)-benzoic acid...)
Affinity DataIC50:  256nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Irreversible type of inhibition)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional

Curated by ChEMBL
LigandPNGBDBM50127980(3-(3-Carboxy-acryloylamino)-benzoic acid | CHEMBL5...)
Affinity DataIC50:  357nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Irreversible type of inhibition)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  360nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164223(2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitr...)
Affinity DataIC50:  420nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164224(CHEMBL192921 | {Imidazo[1,2-d][1,2,4]thiadiazol-3-...)
Affinity DataIC50:  620nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164225(CHEMBL365470 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164226(CHEMBL193724 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  910nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537505(CHEMBL4518615)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164218(CHEMBL192770 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164221(CHEMBL189379 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164219(CHEMBL190568 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537505(CHEMBL4518615)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537506(CHEMBL4574182)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164216(CHEMBL190022 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164222(CHEMBL193212 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164217(CHEMBL192660 | N*1*-Imidazo[1,2-d][1,2,4]thiadiazo...)
Affinity DataIC50:  1.10E+4nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164224(CHEMBL192921 | {Imidazo[1,2-d][1,2,4]thiadiazol-3-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50537506(CHEMBL4574182)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164223(2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitr...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164220(CHEMBL192376 | N-Hexyl-2-nitro-benzenesulfonamide)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164215(2-Nitro-N-[6-(3-nitro-pyridin-2-ylamino)-hexyl]-be...)
Affinity DataIC50:  1.70E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed