TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional
Curated by ChEMBL
Instituto PolitéCnico Nacional
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional
Curated by ChEMBL
Instituto PolitéCnico Nacional
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional
Curated by ChEMBL
Instituto PolitéCnico Nacional
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional
Curated by ChEMBL
Instituto PolitéCnico Nacional
Curated by ChEMBL
Affinity DataIC50: 256nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Irreversible type of inhibition)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional
Curated by ChEMBL
Instituto PolitéCnico Nacional
Curated by ChEMBL
Affinity DataIC50: 357nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Irreversible type of inhibition)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Instituto PolitéCnico Nacional
Curated by ChEMBL
Instituto PolitéCnico Nacional
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibitory activity of the compound against acetylcholinesterase (AChE) from Torpedo californica (Reversible type of inhibition)More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of Wistar rat brain MAOB using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Universidad Aut£Noma Del Estado De Morelos
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of Wistar rat brain MAOA using kynuramine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins ...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research
Curated by ChEMBL
Apotex Research
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair