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Found 51 with Last Name = 'spitler' and Initial = 'jm'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211619((S)-N-(1-(4-(4-ethoxy-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211617((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50172158((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211632((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211636((S)-N-(1-(4-(4-cyclopropyl-2-(2-fluorophenylsulfon...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211605((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  2nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211629((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211627((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211610((S)-N-(1-(4-(4-chloro-2-(pyridin-2-ylsulfonyl)phen...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211604((S)-N-(1-(4-(4-chloro-2-(pyridin-2-ylsulfonyl)phen...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211628((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211609((S)-N-(1-(4-(2-(2-amino-6-fluorophenylsulfonyl)-4-...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211616((S)-N-(1-(4-(4-(cyclopropylamino)-2-(2-fluoropheny...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211620((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211623((S)-N-(1-(4-(4-chloro-2-(2,6-difluorophenylsulfony...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211626((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  7nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211638((S)-N-(1-(4-(4-chloro-2-(cyclohexylsulfonyl)phenyl...)
Affinity DataKi:  8.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211611((S)-N-(1-(4-(4-amino-2-(2-fluorophenylsulfonyl)phe...)
Affinity DataKi:  10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211637((S)-N-(1-(4-(4-chloro-2-(2-(cyclopropylamino)-6-fl...)
Affinity DataKi:  14.4nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211621((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  17nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211630((S)-N-(1-(4-(4-chloro-2-(pyrimidin-2-ylsulfonyl)ph...)
Affinity DataKi:  21nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211614((S)-N-(1-(4-(4-chloro-2-(2-fluoro-6-(methylamino)p...)
Affinity DataKi:  22nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211639((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)p...)
Affinity DataKi:  25nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211618((S)-N-(1-(4-(4-chloro-2-(piperidin-1-ylsulfonyl)ph...)
Affinity DataKi:  58nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211631((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  60.7nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211634((S)-N-(1-(4-(4-chloro-2-(2-(dimethylamino)-6-fluor...)
Affinity DataKi:  115nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211615(CHEMBL245778 | N-((S)-1-{4-[4-chloro-2-(1-oxy-pyri...)
Affinity DataKi:  119nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211622((S)-N-(1-(4-(4-chloro-2-(2-methylfuran-3-ylsulfony...)
Affinity DataKi:  129nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211612((S)-N-tert-butyl-5-chloro-2-(4-(1-(trifluoromethyl...)
Affinity DataKi:  136nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211641((S)-N-(1-(4-(4-chloro-2-(2-fluoro-6-morpholinophen...)
Affinity DataKi:  140nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211613((S)-N-(1-(4-(4-chloro-2-(morpholinosulfonyl)phenyl...)
Affinity DataKi:  192nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211606((S)-N-(1-(4-(4-chloro-2-(quinolin-8-ylsulfonyl)phe...)
Affinity DataKi:  204nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211608((S)-N-(1-(4-(4-chloro-2-(propylsulfonyl)phenylsulf...)
Affinity DataKi:  308nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211640((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211624((S)-5-chloro-N-methyl-2-(4-(1-(methylsulfonamido)e...)
Affinity DataKi:  1.25E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211633((S)-5-chloro-N,N-dimethyl-2-(4-(1-(methylsulfonami...)
Affinity DataKi:  1.27E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211607((S)-5-chloro-2-(4-(1-(methylsulfonamido)ethyl)phen...)
Affinity DataKi:  2.75E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211635((S)-1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)pheny...)
Affinity DataKi:  3.95E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211625((S)-1-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50287485(3-Amino-propane-1-sulfonic acid hydroxy-methyl-ami...)
Affinity DataIC50:  40nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50287486(3-Amino-propane-1-sulfonic acid benzyl-hydroxy-ami...)
Affinity DataIC50:  40nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50087276(3-Amino-propane-1-sulfinic acid (Homohypotaurine) ...)
Affinity DataIC50:  60nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50287484(CHEMBL541547 | [(3-Amino-propane-1-sulfonyl)-hydro...)
Affinity DataIC50:  80nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)
Affinity DataIC50:  200nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50287482(3-Amino-propane-1-sulfonic acid hydroxyamide; hydr...)
Affinity DataIC50:  280nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286226(3-Amino-2-(4-chloro-phenyl)-propane-1-sulfinic aci...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Gamma-aminobutyric acid type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281573(3-Amino-propane-1-sulfonic acid | 3-ammoniopropane...)
Affinity DataIC50:  3.00E+4nMAssay Description:Binding affinity against Gamma-aminobutyric acid type B receptor in rat brain synaptosomes after 30 minutesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286225(3-Amino-2-(4-chloro-phenyl)-propane-1-sulfonic aci...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of Gamma-aminobutyric acid type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286226(3-Amino-2-(4-chloro-phenyl)-propane-1-sulfinic aci...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of Gamma-aminobutyric acid type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286226(3-Amino-2-(4-chloro-phenyl)-propane-1-sulfinic aci...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of Gamma-aminobutyric acid type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
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