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Found 16 with Last Name = 'spreafico' and Initial = 'm'
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50304486((3R,4R,5R,6R)-3-acetamido-6-(acetoxymethyl)tetrahy...)
Affinity DataIC50:  1.13E+5nMAssay Description:Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50077229(CHEMBL300520 | beta-D-galactopyranose | beta-D-gal...)
Affinity DataIC50:  1.05E+6nMAssay Description:Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...More data for this Ligand-Target Pair
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50304487((2R,3R,4S,5S,6R)-2,3,4,5-tetramethoxy-6-(methoxyme...)
Affinity DataIC50:  1.83E+6nMAssay Description:Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50304488((2S,3R,4S,5S,6R)-2,3,4,5-tetramethoxy-6-(methoxyme...)
Affinity DataIC50:  2.83E+6nMAssay Description:Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50240803(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Affinity DataIC50: >3.00E+7nMAssay Description:Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50304486((3R,4R,5R,6R)-3-acetamido-6-(acetoxymethyl)tetrahy...)
Affinity DataKd:  1.50E+5nMAssay Description:Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50077229(CHEMBL300520 | beta-D-galactopyranose | beta-D-gal...)
Affinity DataKd:  1.46E+6nMAssay Description:Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...More data for this Ligand-Target Pair
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50304487((2R,3R,4S,5S,6R)-2,3,4,5-tetramethoxy-6-(methoxyme...)
Affinity DataKd:  2.20E+6nMAssay Description:Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50304488((2S,3R,4S,5S,6R)-2,3,4,5-tetramethoxy-6-(methoxyme...)
Affinity DataKd:  2.76E+6nMAssay Description:Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50240803(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Affinity DataKd: >1.00E+7nMAssay Description:Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327100(CHEMBL1254194 | sodium(1R,3R,4R,5S)-5-acetamido-1-...)
Affinity DataKd: >8.00E+5nMAssay Description:Binding affinity to mouse MAGd1-3Fc domain expressed in CHO-Lec1 cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327099(CHEMBL1253679 | sodium2R,4S,5R,6R)-6-((1R,2R)-3-(4...)
Affinity DataKd:  500nMAssay Description:Binding affinity to mouse MAGd1-3Fc domain expressed in CHO-Lec1 cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.60E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc domain expressed in CHO-Lec1 cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50292880(2-(Trimethylsilyl)ethyl (Sodium 5-Acetamido-9-benz...)
Affinity DataKd:  3.26E+4nMAssay Description:Binding affinity to human IgG Fc-domain tagged MAG N-terminal domain expressed in CHO cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50292878((Sodium 5-Acetamido-9-(4-chlorobenzamido)-3,5,9-tr...)
Affinity DataKd:  2.83E+3nMAssay Description:Binding affinity to human IgG Fc-domain tagged MAG N-terminal domain expressed in CHO cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50292879((Sodium 5-Acetamido-9-benzamido-3,5,9-trideoxy-D-g...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to human IgG Fc-domain tagged MAG N-terminal domain expressed in CHO cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed