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Found 44 with Last Name = 'spyrakis' and Initial = 'f'
TargetThymidylate synthase(Homo sapiens (Human))
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50590309(CHEMBL5196526)
Affinity DataKi:  4.00E+4nMAssay Description:Non competitive type inhibition of human TS assessed as inhibition constant using varying levels of mTHF as substrate by UV-Vis spectroscopy based an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of human recombinant serine racemase expressed in Escherichia coli Rosetta 2 (DE3) cells using L-serine as substrate by horseradish peroxi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  6.60E+4nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50590310(CHEMBL5195943)
Affinity DataKi:  7.30E+4nMAssay Description:Non competitive type inhibition of human TS assessed as inhibition constant using varying levels of mTHF as substrate by UV-Vis spectroscopy based an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119563(CHEBI:45969 | TRICARBALLYLIC ACID)
Affinity DataKi:  1.30E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119562(CHEMBL3617724)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119565(CHEMBL3617722)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119564(CHEMBL3617723)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119560(CHEMBL3617727)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine racemase(Homo sapiens (Human))
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50119561(CHEMBL3617725)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593724(CHEMBL5194388)
Affinity DataIC50:  69nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593730(CHEMBL5172658)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50509767(CHEMBL4513510)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 assessed as reduction in NADPH-dependent 9,10-phenanthrenequinone convers...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50509981(CHEMBL3990606)
Affinity DataIC50:  134nMAssay Description:Inhibition of CSNK1D (unknown origin) using CSNK1D/Ser/Thr 11 peptide incubated for 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593732(CHEMBL5174744)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593726(CHEMBL5204156)
Affinity DataIC50:  210nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593727(CHEMBL5170149)
Affinity DataIC50:  220nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593728(CHEMBL5170401)
Affinity DataIC50:  260nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593729(CHEMBL5175151)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593725(CHEMBL5206583)
Affinity DataIC50:  310nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50277998(CHEMBL4174786)
Affinity DataIC50:  310nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50509984(CHEMBL4476186)
Affinity DataIC50:  354nMAssay Description:Inhibition of CSNK1D (unknown origin) using CSNK1D/Ser/Thr 11 peptide incubated for 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593722(CHEMBL5191752)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593723(CHEMBL5187723)
Affinity DataIC50:  470nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50509983(CHEMBL3940534)
Affinity DataIC50:  848nMAssay Description:Inhibition of CSNK1D (unknown origin) using CSNK1D/Ser/Thr 11 peptide incubated for 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50509982(CHEMBL4519384)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of CSNK1D (unknown origin) using CSNK1D/Ser/Thr 11 peptide incubated for 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50593731(CHEMBL5183881)
Affinity DataIC50:  1.63E+3nMAssay Description:Inhibition of recombinant human AKR1C3 transfected in Escherichia coli BL21 (DE) assessed as reduction in NADPH production using S-tetralol as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50509767(CHEMBL4513510)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant human AKR1C2 transfected in Escherichia coli BL21 assessed as reduction in NADPH-dependent 9,10-phenanthrenequinone convers...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423697(CHEMBL568986)
Affinity DataKd:  6.03E+4nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423698(CHEMBL568987)
Affinity DataKd:  1.91E+5nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50590310(CHEMBL5195943)
Affinity DataKd:  1.20E+5nMAssay Description:Mixed type inhibition of human TS assessed as inhibitor dissociation constant by measuring changes in slope of the double reciprocal plot using dTMP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetThymidylate synthase(Homo sapiens (Human))
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50590309(CHEMBL5196526)
Affinity DataKd:  4.40E+4nMAssay Description:Mixed type inhibition of human TS assessed as inhibitor dissociation constant by measuring changes in slope of the double reciprocal plot using dTMP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423699(CHEMBL571766)
Affinity DataKd:  5.75E+5nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423700(CHEMBL568812)
Affinity DataKd:  1.02E+6nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423701(CHEMBL576268)
Affinity DataKd:  2.29E+6nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423702(CHEMBL585737)
Affinity DataKd:  3.39E+6nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423703(CHEMBL582831)
Affinity DataKd:  3.31E+6nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423704(CHEMBL567022)
Affinity DataKd:  7.08E+6nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423705(CHEMBL569309)
Affinity DataKd:  1.32E+7nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423706(CHEMBL570451)
Affinity DataKd:  1.51E+7nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423707(CHEMBL571997)
Affinity DataKd:  4.37E+4nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423709(CHEMBL568900)
Affinity DataKd:  2.51E+4nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423710(CHEMBL569308)
Affinity DataKd:  3.89E+4nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine synthase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
University Of Parma

Curated by ChEMBL
LigandPNGBDBM50423708(CHEMBL568828)
Affinity DataKd:  2.57E+4nMAssay Description:Binding affinity to Haemophilus influenzae O-acetylserine sulfhydrylase expressed in Escherichia coli BL21 (DE3) by fluorescence emission spectra ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed