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Found 25 with Last Name = 'srinivasa rao' and Initial = 'a'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM22369(4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofu...)
Affinity DataIC50:  57nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124787(2-(5-Methoxy-1H-benzoimidazol-2-ylsulfanylmethyl)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124792(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-benzothi...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124790(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-1H-benzoi...)
Affinity DataIC50:  1.47E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124793(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-5-nitro-...)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124788(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-5-methyl...)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124782(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-benzooxa...)
Affinity DataIC50:  2.77E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124786(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-5-methoxy...)
Affinity DataIC50:  6.25E+3nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124789(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-benzothia...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124796(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-5-methyl-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124795(5-Methoxy-2-(2-methoxy-6-pentadecyl-benzylsulfanyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124794(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-1H-benzo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124791(5-Difluoromethoxy-2-(2-methoxy-6-pentadecyl-benzyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124784(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-benzooxaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124783(5-Difluoromethoxy-2-(2-ethoxy-6-pentadecyl-benzyls...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM22369(4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofu...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124787(2-(5-Methoxy-1H-benzoimidazol-2-ylsulfanylmethyl)-...)
Affinity DataIC50:  3.84E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124785(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-5-nitro-1...)
Affinity DataIC50:  3.84E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 in human whole blood assay as LPS induced PGE-2 generation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124790(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-1H-benzoi...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124792(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-benzothi...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124785(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-5-nitro-1...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124782(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-benzooxa...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124793(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-5-nitro-...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124786(2-(2-Ethoxy-6-pentadecyl-benzylsulfanyl)-5-methoxy...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Vittal Mallya Scientific Research Foundation

Curated by ChEMBL
LigandPNGBDBM50124788(2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-5-methyl...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 in human whole blood assay as TXB2 generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed