Compile Data Set for Download or QSAR
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Found 61 with Last Name = 'stachew' and Initial = 'cf'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133557(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-morphol...)
Affinity DataKi:  500nMAssay Description:Inhibition of Tau Protein Kinase II (TPK II)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133573(CHEMBL119530 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  900nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133579(CHEMBL117950 | N-(tert-butoxy)-N'-[2-(2,6-dichloro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133557(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-morphol...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133575(CHEMBL119041 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  3.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133564(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-pyrroli...)
Affinity DataIC50:  3.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133551(CHEMBL119143 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  4.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133569(1-Morpholin-4-yl-3-[2-(pyridine-2-sulfonylmethyl)-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133580(CHEMBL119796 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  5.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133566(CHEMBL117778 | N-{2-[(methylsulfonyl)methyl]-1,3-t...)
Affinity DataIC50:  6.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133555(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-piperid...)
Affinity DataIC50:  6.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133567(CHEMBL118685 | N-(allyloxy)-N'-[2-(2,6-dichloroben...)
Affinity DataIC50:  6.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133556(1-Morpholin-4-yl-3-(2-phenyl-thiazol-4-yl)-urea | ...)
Affinity DataIC50:  6.00E+3nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133576(CHEMBL116615 | N-phenoxy-N'-(2-phenyl-1,3-thiazol-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133556(1-Morpholin-4-yl-3-(2-phenyl-thiazol-4-yl)-urea | ...)
Affinity DataIC50:  9.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133549(CHEMBL117800 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  9.00E+3nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133574(1-Azepan-1-yl-3-[2-(2,6-dichloro-benzyl)-thiazol-4...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133565(CHEMBL116339 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133551(CHEMBL119143 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133568(1-[2-(2-Chloro-phenyl)-thiazol-4-yl]-3-morpholin-4...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133569(1-Morpholin-4-yl-3-[2-(pyridine-2-sulfonylmethyl)-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133557(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-morphol...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133559(1-Morpholin-4-yl-3-(2-thiophen-2-yl-thiazol-4-yl)-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133579(CHEMBL117950 | N-(tert-butoxy)-N'-[2-(2,6-dichloro...)
Affinity DataIC50:  1.50E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133560(CHEMBL117779 | N-[2-(3-methylphenyl)-1,3-thiazol-4...)
Affinity DataIC50:  1.60E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133553(1-Morpholin-4-yl-3-(2-m-tolyl-thiazol-4-yl)-urea |...)
Affinity DataIC50:  2.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133580(CHEMBL119796 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  2.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133552(CHEMBL325452 | N-(2-benzyl-1,3-thiazol-4-yl)-N'-ph...)
Affinity DataIC50:  2.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133550(1-[2-(4-Methoxy-phenoxymethyl)-thiazol-4-yl]-3-mor...)
Affinity DataIC50:  2.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133564(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-pyrroli...)
Affinity DataIC50:  2.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133577(1-Morpholin-4-yl-3-(2-phenylsulfanylmethyl-thiazol...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133559(1-Morpholin-4-yl-3-(2-thiophen-2-yl-thiazol-4-yl)-...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133577(1-Morpholin-4-yl-3-(2-phenylsulfanylmethyl-thiazol...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133568(1-[2-(2-Chloro-phenyl)-thiazol-4-yl]-3-morpholin-4...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133553(1-Morpholin-4-yl-3-(2-m-tolyl-thiazol-4-yl)-urea |...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133550(1-[2-(4-Methoxy-phenoxymethyl)-thiazol-4-yl]-3-mor...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133555(1-[2-(2,6-Dichloro-benzyl)-thiazol-4-yl]-3-piperid...)
Affinity DataIC50:  3.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133576(CHEMBL116615 | N-phenoxy-N'-(2-phenyl-1,3-thiazol-...)
Affinity DataIC50:  3.50E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133567(CHEMBL118685 | N-(allyloxy)-N'-[2-(2,6-dichloroben...)
Affinity DataIC50:  4.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133554(1-(2-Benzyl-thiazol-4-yl)-3-morpholin-4-yl-urea | ...)
Affinity DataIC50:  5.50E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133565(CHEMBL116339 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  6.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133574(1-Azepan-1-yl-3-[2-(2,6-dichloro-benzyl)-thiazol-4...)
Affinity DataIC50:  7.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133561(1-Morpholin-4-yl-3-(2-phenoxymethyl-thiazol-4-yl)-...)
Affinity DataIC50:  8.00E+4nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133566(CHEMBL117778 | N-{2-[(methylsulfonyl)methyl]-1,3-t...)
Affinity DataIC50:  9.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133575(CHEMBL119041 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50:  9.00E+4nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133573(CHEMBL119530 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133582(1-Morpholin-4-yl-3-(2-p-tolyl-thiazol-4-yl)-urea |...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133563(1-(2-Ethyl-thiazol-4-yl)-3-morpholin-4-yl-urea | C...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133581(1-[2-(4-Chloro-phenyl)-thiazol-4-yl]-3-morpholin-4...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to inhibit Cyclin-dependent kinase 5-p35.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50133549(CHEMBL117800 | N-[2-(2,6-dichlorobenzyl)-1,3-thiaz...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to inhibit cyclin-dependent kinase 2-cyclin A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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