Affinity DataKi: 0.450nMAssay Description:Inhibition of binding to membranes from HEK293 cells expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Binding affinity for Adenosine A1 receptor of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Inhibition of binding to membranes from HEK293 cells expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for Adenosine A1 receptor from Guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.56nMAssay Description:Binding affinity for Adenosine A1 receptor from Guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.56nMAssay Description:Binding affinity for Adenosine A1 receptor from Guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity for Adenosine A1 receptor from Guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.93nMAssay Description:Binding affinity for Adenosine A1 receptor from Guinea pig membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.77nMAssay Description:Binding affinity for Adenosine A1 receptor of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 5.12nMAssay Description:Binding affinity for Adenosine A1 receptor of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity for Adenosine A1 receptor of rat forebrainMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to bovine serum albuminMore data for this Ligand-Target Pair
TargetSterol carrier protein 2(Homo sapiens (Human))
European Molecular Biology Laboratory
Curated by ChEMBL
European Molecular Biology Laboratory
Curated by ChEMBL
Affinity DataKd: 339nMAssay Description:Binding affinity to site 1 of human mature SCP2More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Binding affinity to bovine serum albuminMore data for this Ligand-Target Pair
TargetSterol carrier protein 2(Homo sapiens (Human))
European Molecular Biology Laboratory
Curated by ChEMBL
European Molecular Biology Laboratory
Curated by ChEMBL
Affinity DataKd: 947nMAssay Description:Binding affinity to site 2 of human mature SCP2More data for this Ligand-Target Pair